2023 - epigenetics modulation frontier

Hydrocortisone 21-octanoate-d4

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Hydrocortisone 21-octanoate-d4 Biological Activity：Hydrocortisone 21-octanoate-d4 is the deuterium labeled Hydrocortisone 21-octanoate. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | […]

MTH-DL-Tyrosine

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. MTH-DL-Tyrosine CAS No. : 886-26-0 Biological Activity：MTH-DL-Tyrosine is a tyrosine derivative. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | […]

(R)-Elagolix

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. (R)-Elagolix CAS No. : 834153-87-6 Biological Activity：Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). Target: GnRH in vitro: Elagolix is a short-acting, nonpeptide, GnRH antagonist, administered orally, that unlike injectable depot GnRH agonists […]

Mastoparan

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Mastoparan CAS No. : 72093-21-1 Biological Activity：Mastoparan, a tetradecapeptide which is a component of wasp venom, stimulates release of prolactin from cultured rat anterior pituitary cells. Research Area：Metabolic Disease Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione […]

dTAGV-1-NEG

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. dTAGV-1-NEG CAS No. : 2451573-87-6 Biological Activity：dTAGV-1-NEG is a diastereomer and as a heterobifunctional negative control of dTAGV-1. dTAGV-1 is an FKBP12F36V-selective degrader. Research Area：Cancer Targets：FKBP|PROTACs Related Small Molecules:PROTAC Sirt2 Degrader-1;DB0614;PROTAC VEGFR-2 degrader-2;CCT367766 formic;HDAC6 degrader-1;SAFit2;PROTAC Axl Degrader 2;PhosTAC7;MS98;JPS014;PROTAC PARP1 degrader;MD-224;FKBP12 PROTAC dTAG-7;SJ10542;MS8815;RIP2 Kinase Inhibitor 4;PROTAC […]

CIQ

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. CIQ CAS No. : 486427-17-2 Biological Activity：CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. Research Area：Neurological Disease Targets：iGluR Related Screening Libraries:Bioactive Compound Library Plus;Membrane Transporter/Ion Channel Compound Library;Neuronal Signaling Compound Library;Neurotransmitter Receptor Compound Library; Related Small Molecules:Quinolinic acid-d3;1-Aminocyclobutanecarboxylic acid;Glycine-1-13C,15N;ZL006;PYD-106;NMDA-IN-2;JAMI1001A;(S)-Willardiine;Fanapanel;(S)-AMPA;L-Glutamic […]

RIPA-56

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. RIPA-56 CAS No. : 1956370-21-0 Biological Activity：RIPA-56 is a highly potent, selective, and metabolically stable inhibitor of receptor-interacting protein 1 (RIP1) with an IC50 of 13 nM. RIPA-56 can be used for the treatment of systemic inflammatory response syndrome. Research Area：Inflammation/Immunology Targets：RIP kinase Related Screening […]

CFTR corrector 8

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. CFTR corrector 8 CAS No. : 1918142-35-4 Biological Activity：CFTR corrector 8 is a potent CFTR modulator. CFTR can be used in the research of cystic fibrosis. Research Area：Inflammation/Immunology Targets：CFTR Related Small Molecules:PG01;CP-628006;SRI-37240;Urocortin III (mouse) (free acid);NJH-2-056;Elexacaftor;GlyH-101;Cavosonstat;Kobusin;GLPG1837;(R)-Posenacaftor sodium;GLPG2451;CFTR corrector 9;CFTR corrector 2;Vanzacaftor;CFTR corrector 4;Posenacaftor sodium;NJH-2-057;KM11060;Nesolicaftor;Galicaftor;Tezacaftor;PPQ-102;SRI-41315;CFTR corrector […]

Edrophonium chloride

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Edrophonium chloride CAS No. : 116-38-1 Biological Activity：Edrophonium chloride is a readily reversible acetylcholinesterase inhibitor; prevents breakdown of the neurotransmitter acetylcholine and acts by competitively inhibiting the enzyme acetylcholinesterase, mainly at the neuromuscular junction. Research Area：Neurological Disease Targets：Cholinesterase (ChE) Related Screening Libraries:Drug Repurposing Compound Library […]

LSD1/ER-IN-1

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. LSD1/ER-IN-1 Biological Activity：LSD1/ER-IN-1 (compound 11g) is a potent ER and LSD1 inhibitor, with an IC50 of 1.55 μM (LSD1). LSD1/ER-IN-1 has high affinity selectivity for ERα protein, with α/β ratio of 7.11. LSD1/ER-IN-1 shows good antiproliferative activity against MCF-7 breast cancer cells, with an IC50 […]