Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. GSK2018682 CAS No. : 1034688-30-6 Biological Activity：GSK2018682 is an agonist for S1P1 and S1P5 receptor with pEC50s of 7.7 and 7.2, respectively, and has no agonist activity towards human S1P2, S1P3, or S1P4. GSK2018682 is used in the research of multiple sclerosis. Research Area：Inflammation/Immunology Targets：LPL […]
For research use only. We do not sell to patients. Pregnanetriol 3α-O-β-D-glucuronide-d4 Biological Activity：Pregnanetriol 3α-O-β-D-glucuronide-d4 is the deuterium labeled Pregnanetriol 3α-O-β-D-glucuronide. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | […]
For research use only. We do not sell to patients. Ciclopirox-d11 Biological Activity：Ciclopirox-d11 (HOE296b-d11) is the deuterium labeled Ciclopirox. Ciclopirox (HOE296b) is a synthetic antifungal agent that can be used for superficial mycoses reseaech. Ciclopirox olamine has a very broad spectrum of activity and inhibits dermatophytes, yeasts, molds, and many Gram-positive and Gram-negative species pathogenic. […]
For research use only. We do not sell to patients. Mangiferin CAS No. : 4773-96-0 Biological Activity：Mangiferin is a Nrf2 activator. Mangiferin suppresses nuclear translocation of the NF-κB subunits p65 and p50. Mangiferin exhibits antioxidant, antidiabetic, antihyperuricemic, antiviral, anticancer and antiinflammatory activities[2][3]. Research Area：Cancer Targets：Keap1-Nrf2|NF-κB|Apoptosis Related Screening Libraries:Natural Product Library Plus;Bioactive Compound Library Plus;Apoptosis Compound […]
For research use only. We do not sell to patients. Thalidomide-NH-amido-C6-NH2 hydrochloride Biological Activity：Thalidomide-NH-amido-C6-NH2 hydrochloride is a synthesized E3 ligase ligand-linker conjugate that incorporates the Thalidomide based cereblon ligand and a linker used in PROTAC technology. Research Area：Cancer Targets：E3 Ligase Ligand-Linker Conjugates Related Small Molecules:cIAP1 Ligand-Linker Conjugates 6 hydrochloride;(S,R,S)-AHPC-Me-C10-NH2;cIAP1 Ligand-Linker Conjugates 2;Glutarimide-Isoindolinone-NH-PEG3-COOH;cIAP1 Ligand-Linker Conjugates 4;(S,R,S)-AHPC-Me-C7 […]
For research use only. We do not sell to patients. D-Lin-MC3-DMA CAS No. : 1224606-06-7 Biological Activity：D-Lin-MC3-DMA, an ionizable cationic lipid, is a potent siRNA delivery vehicle. Research Area：Cancer Targets：Others Related Screening Libraries:Bioactive Compound Library Plus;Anti-Cancer Compound Library; Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant […]
For research use only. We do not sell to patients. Imidafenacin CAS No. : 170105-16-5 Biological Activity：Imidafenacin(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM). IC50 value: 0.3 nM(M3) [1] in vitro: KRP-197 showed equipotent anti-M2 and anti-M3 activity and decreased subtype-selectivity […]
For research use only. We do not sell to patients. Zandatrigine CAS No. : 2154406-04-7 Biological Activity：Zandatrigine (NBI-921352) is a sodium channel protein type 8 subunit alpha (Scn8α) blocker. Research Area：Neurological Disease Targets：Sodium Channel Related Screening Libraries:Drug Repurposing Compound Library Plus; Clinical Compound Library Plus;Bioactive Compound Library Plus;Membrane Transporter/Ion Channel Compound Library;Clinical Compound Library;Drug Repurposing […]
For research use only. We do not sell to patients. Diltiazem hydrochloride CAS No. : 33286-22-5 Biological Activity：Diltiazem hydrochloride is a Ca2+ influx inhibitor (slow channel blocker or calcium antagonist). Research Area：Cardiovascular Disease Targets：Calcium Channel Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;Membrane Transporter/Ion Channel Compound Library;Neuronal […]
For research use only. We do not sell to patients. Cambinol CAS No. : 14513-15-6 Biological Activity：Cambinol is a SIRT1 and SIRT2 inhibitor with IC50 values of 56 μM and 59 μM, respectively. Cambinol is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor (exosome inhibitor)[2]. Research Area：Cancer Targets：Sirtuin|Apoptosis|Phospholipase Related Screening Libraries:Bioactive Compound Library Plus;Apoptosis Compound […]