Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. BQ-788 CAS No. : 173326-37-9 Biological Activity：BQ-788 is a potent, selective ETB receptor antagonist with IC50 of 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells, poorly inhibiting the binding to ETA receptors in human neuroblastoma cell line SK-N-MC cells with IC50 […]
For research use only. We do not sell to patients. Pomalidomide-amido-C4-amido-PEG2-C2-NH-Boc CAS No. : 2435720-04-8 Biological Activity：Pomalidomide-amido-C4-amido-PEG2-C2-NH-Boc is a synthesized E3 ligase ligand-linker conjugate that incorporates the Pomalidomide based cereblon ligand and 2-unit PEG linker used in PROTAC technology. Research Area：Cancer Targets：E3 Ligase Ligand-Linker Conjugates Related Small Molecules:cIAP1 Ligand-Linker Conjugates 6 hydrochloride;(S,R,S)-AHPC-Me-C10-NH2;cIAP1 Ligand-Linker Conjugates 2;Glutarimide-Isoindolinone-NH-PEG3-COOH;cIAP1 […]
For research use only. We do not sell to patients. Todralazine CAS No. : 14679-73-3 Biological Activity：Todralazine (Ecarazine) is an anti-hypertensive agent, acts as a β2AR blocker, with antioxidant and free radical scavenging activity. Research Area：Cardiovascular Disease|Endocrinology Targets：Adrenergic Receptor Related Small Molecules:ARC 239 dihydrochloride;Yohimbine;Glaucine;Salbutamol;BI-167107;Talibegron hydrochloride;Arotinolol;SR59230A;Higenamine hydrochloride;Navafenterol saccharinate;Isoprenaline hydrochloride;Bevantolol;Zilpaterol-d7;Ritanserin;A55453;Povafonidine;β3-AR agonist 1;Tulobuterol;AGN 192836;KUC-7322;Oxyfedrine;Urapidil hydrochloride;Detomidine hydrochloride;Oxprenolol-d7 hydrochloride;Nicergoline;Synephrine hemitartrate;ADRA1D […]
For research use only. We do not sell to patients. ST-193 hydrochloride CAS No. : 2320274-72-2 Biological Activity：ST-193 hydrochloride is a potent broad-spectrum arenavirus inhibitor; inhibits Guanarito, Junin, Lassa and Machupo virus with IC50 values of 0.44, 0.62, 1.4 and 3.1 nM, respectively. Research Area：Infection Targets：Arenavirus Related Screening Libraries:Bioactive Compound Library Plus;Anti-Infection Compound Library; Antiviral […]
For research use only. We do not sell to patients. DS20362725 CAS No. : 2735803-20-8 Biological Activity：DS20362725 is an estrogen-related receptor α (ERRα) agonist. DS20362725 inhibits the binding between receptor-interacting protein 140 (RIP140) corepressor peptide (10 nM) and GST-ERRα ligand-binding domain (LBD; 1.2 μM) with an IC50 value of 0.6 μM. DS20362725 can be used […]
For research use only. We do not sell to patients. Drinidene CAS No. : 53394-92-6 Biological Activity：Drinidene can be used for the research of pain disorders extracted from patent AU2018254530A1. Research Area：Neurological Disease Targets：Others Related Screening Libraries:Bioactive Compound Library Plus; Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione […]
For research use only. We do not sell to patients. CCG-50014 CAS No. : 883050-24-6 Biological Activity：CCG-50014 is the most potent against the regulator of G-protein signaling protein type 4 (RGS4) (IC50 =30 nM) and is >20-fold selective for RGS4 over other RGS proteins. CCG-50014 binds covalently to the RGS, forming an adduct on two […]
For research use only. We do not sell to patients. Kanamycins sulfate CAS No. : 70560-51-9 Biological Activity：Kanamycins sulfate is a broad-spectrum antibiotic, can be used in certain severe staphylococcal or Gram-negative bacillary infections. Kanamycin sulfate has certain ototoxicity[2]. Research Area：Infection Targets：Bacterial|Antibiotic Related Small Molecules:Sandramycin;LLO (91-99);Gepotidacin;Oritavancin;Monascorubrin;Azlocillin sodium salt;Herbimycin A;Antibacterial agent 45;Leucomycin;Isouvaretin;Antibacterial agent 99;Vidarabine monohydrate;Nafcillin;Antitubercular agent-28;Ochromycinone;Staurosporine;Nucleocidin;(±)-Leucine-13C-1;Ciclopirox-d11;Ciclopirox […]
For research use only. We do not sell to patients. Busulfan CAS No. : 55-98-1 Biological Activity：Busulfan is a potent alkylating antineoplastic agent. Busulfan causes DNA damage by cross-linking DNAs and DNA and proteins. Busulfan inhibits thioredoxin reductase. Busulfan induces apoptosis. Busulfan is an immunosuppressive and myeloablative chemotherapeutic drug[2][3]. Research Area：Cancer|Inflammation/Immunology Targets：DNA Alkylator/Crosslinker|Apoptosis Related Screening […]
For research use only. We do not sell to patients. EEDi-5285 CAS No. : 2488952-40-3 Biological Activity：EEDi-5285 is an exceptionally potent and orally active embryonic ectoderm development (EED) inhibitor with an IC50 value of 0.2 nM for binds to the EED protein. EEDi-5285 has anti-cancer activity. Research Area：Cancer Targets：Histone Methyltransferase Related Screening Libraries:Bioactive Compound Library […]