Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. Cytarabine-d2 CAS No. : 40632-26-6 Biological Activity：Cytarabine-d2 is the deuterium labeled Cytarabine. Cytarabine, a nucleoside analog, causes S phase cell cycle arrest and inhibits DNA polymerase. Cytarabine inhibits DNA synthesis with an IC50 of 16 nM. Cytarabine has antiviral effects against HSV[2]. Research Area：Cancer|Infection Targets：HSV|Nucleoside […]
For research use only. We do not sell to patients. Cathepsin G Inhibitor I CAS No. : 429676-93-7 Biological Activity：Cathepsin G Inhibitor I is a potent, selective, reversible, competitive, non-peptide inhibitor of cathepsin G. Research Area：Inflammation/Immunology Targets：Cathepsin Related Screening Libraries:Bioactive Compound Library Plus;Immunology/Inflammation Compound Library;Metabolism/Protease Compound Library;Angiogenesis-Related Compound Library; Related Small Molecules:Calpeptin;Gly-Phe-β-naphthylamide;Z-FY-CHO;Balicatib;Cathepsin D and E […]
For research use only. We do not sell to patients. Magnesium silicate CAS No. : 1343-88-0 Biological Activity：Magnesium silicate (Activated magnesium silicate) is a compound of magnesium oxide (MgO) and silicon dioxide (SiO2). Magnesium silicate is used in antiacid and antiulcer preparation, and as a deodorizer, decolorizer and antifungal. Research Area：Infection|Inflammation/Immunology Targets：Fungal Related Screening Libraries:Bioactive […]
For research use only. We do not sell to patients. (Rac)-MEM 1003 CAS No. : 165187-25-7 Biological Activity：(Rac)-MEM 1003 is the racemate of MEM 1003. MEM 1003, a dihydropyridine compound, is a potent L-type Ca2+ channel antagonist and has the potential for Alzheimer’s disease research. Research Area：Others Targets：Calcium Channel Related Screening Libraries:Bioactive Compound Library Plus;Membrane […]
For research use only. We do not sell to patients. Pneumadin, rat CAS No. : 130918-90-0 Biological Activity：Pneumadin, rat (PNM) is a decapeptide, which possess a potent stimulating effect on arginine-vasopressin (AVP) release. Pneumadin, rat (PNM) exerts a marked antidiuretic effect in animals with functional AVP system[2]. Research Area：Metabolic Disease Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 […]
For research use only. We do not sell to patients. SN 6 CAS No. : 415697-08-4 Biological Activity：SN 6 is a selective Na+/Ca2+ exchanger (NCX) inhibitor, and inhibits 45Ca2+ uptake by NCX1, NCX2, and NCX3, with IC50s of 2.9, 16, and 8.6 μM, respectively. Research Area：Cardiovascular Disease Targets：Na+/Ca2+ Exchanger Related Screening Libraries:Bioactive Compound Library Plus;Membrane […]
For research use only. We do not sell to patients. Giredestrant CAS No. : 1953133-47-5 Biological Activity：Giredestrant (GDC-9545), a non-steroidal estrogen receptor (ER) ligand, is an orally active and selective ER antagonist. Giredestrant potently competes with Estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity. Research […]
For research use only. We do not sell to patients. NOS-IN-3 CAS No. : 2761725-68-0 Biological Activity：NOS-IN-3 (Compound 9a) is a potent, selective, imidamide derived NOS inhibitor with an IC50 against iNOS of 4.6 µM, without inhibiting eNOS. NOS-IN-3 has little toxicity and can be studied in the treatment of inducible isoform involved diseases, such […]
For research use only. We do not sell to patients. 3,29-Dibenzoyl rarounitriol CAS No. : 873001-54-8 Biological Activity：3,29-Dibenzoyl rarounitriol is one major bioactive compound of multiflorane triterpene esters Trichosanthes kirilowii, can be chosen as the marker for quantitation of Trichosanthes kirilowii. Research Area：Others Targets：Others Related Screening Libraries:Natural Product Library Plus;Bioactive Compound Library Plus;Natural Product Library;Terpenoids […]
For research use only. We do not sell to patients. SWE101 CAS No. : 2376322-12-0 Biological Activity：SWE101 (compound 22 b) is a potent soluble epoxide hydrolase (sEH)-P inhibitor with IC50s of 4 μM and 2.8 μM for human and rat sEH-P, respectively. SWE101 does not inhibit neither hydrolase nor phosphatase activity of the mouse sEH. […]