Giredestrant

For research use only. We do not sell to patients.

Giredestrant

CAS No. : 1953133-47-5

Biological Activity:Giredestrant (GDC-9545), a non-steroidal estrogen receptor (ER) ligand, is an orally active and selective ER antagonist. Giredestrant potently competes with Estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity.

Research Area:Cancer

Targets:Estrogen Receptor/ERR

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