Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. Gefapixant citrate CAS No. : 2310299-91-1 Biological Activity：Gefapixant citrate is an orally active and potent purinergic P2X3 receptor (P2X3R) antagonist, with IC50 values of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. Gefapixant citrate can be used for the research […]
For research use only. We do not sell to patients. RORγt inverse agonist 30 CAS No. : 1445901-41-6 Biological Activity：RORγt inverse agonist 30 (Compound 1) is a potent RORγt inverse agonist with the IC50 of 46 nM. Targeting the nuclear receptor RORγt is effective in autoimmune disorders. Research Area：Inflammation/Immunology Targets：ROR Related Small Molecules:RORγt inhibitor 1;GNE-6468;SR3335;GNE-0946;RORγt […]
For research use only. We do not sell to patients. SI-2 hydrochloride CAS No. : 1992052-49-9 Biological Activity：SI-2 (EPH 116 hydrochloride) is a highly promising SRC-3 inhibitor (PPI), with IC50 values of 3-20 nM for breast cancer cell death. SI-2 (EPH 116 hydrochloride) has a much improved toxicity and pharmacokinetic profile, with acceptable oral availability. […]
For research use only. We do not sell to patients. (S)-MCPG CAS No. : 150145-89-4 Biological Activity：(S)-MCPG ((+)-MCPG) is a potent group I/II metabotropic glutamate receptor (mGluRs) antagonist and the active isomer of (RS)-MCPG (HY-100371). (S)-MCPG can be used for the study of the function of mGluRs in spatial learning[2]. Research Area：Neurological Disease Targets：mGluR Related […]
For research use only. We do not sell to patients. Human IgG2 kappa, Isotype Control Biological Activity：Human IgG2 kappa, Isotype Control, a human monoclonal antibody, is an isotype control for human IgG2κ antibody. Research Area：Inflammation/Immunology Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | […]
For research use only. We do not sell to patients. t-Boc-N-amido-PEG6-Tos CAS No. : 1264015-76-0 Biological Activity：t-Boc-N-amido-PEG6-Tos is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs. Research Area：Cancer Targets：PROTAC Linkers Related Small Molecules:N-(Mal-PEG6)-N-bis(PEG7-TCO);Propargyl-PEG2-CH2COOH;NHS ester-PEG10-COOH;Tos-PEG5-Boc;Bis-PEG6-NHS ester;Azide-PEG12-alcohol;Fmoc-PEG6-NHS ester;Boc-C1-PEG3-C4-OBn;Boc-NH-PEG8-C2-Br;Propargyl-PEG14-Boc;m-PEG21-OH;Bromo-PEG3-THP;m-PEG8-Ms;Bis-PEG10-NHS ester;TCO-PEG3-acid;m-PEG8-DBCO;Azide-PEG6-Tos;Acid-PEG3-C2-Boc;m-PEG-mal (MW 2000);Benzyl-PEG7-t-butyl ester;Boc-Pip-alkyne-Ph-COOH;Biotin-PEG2-C6-azide;Bis-PEG4-acid;Active-mono-sulfone-PEG8-acid;Br-PEG6-C2-NHBoc;HO-PEG8-CH2COOH;NH2-PEG4-CH2CH2COOH;N-(Propargyl-PEG2)-N-Boc-PEG3-t-butyl ester;Bromoacetamido-PEG8-Boc;Carboxy-PEG2-sulfonic acid Trending products：Recombinant Proteins | Bioactive Screening Libraries | […]
For research use only. We do not sell to patients. GW842166X CAS No. : 666260-75-9 Biological Activity：GW842166X is a potent and selective cannabinoid receptor 2 (CB2) agonist with IC50 values of 63 and 91 nM for human and rat CB2, respectively. Research Area：Inflammation/Immunology|Neurological Disease Targets：Cannabinoid Receptor Related Screening Libraries:Covalent Screening Library Plus;Clinical Compound Library Plus;Bioactive […]
For research use only. We do not sell to patients. Herbacetin-3-sophoroside-8–glucoside CAS No. : 77298-68-1 Biological Activity：Herbacetin-3-sophoroside-8–glucoside is a natural product that can be isolated from Equisetum hyemale. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural […]
For research use only. We do not sell to patients. SNS-032 CAS No. : 345627-80-7 Biological Activity：SNS-032 (BMS-387032) is a potent and selective inhibitor of CDK2, CDK7, and CDK9 with IC50s of 38 nM, 62 nM and 4 nM, respectively. SNS-032 has antitumor effect. Research Area：Cancer Targets：CDK|Apoptosis Related Screening Libraries:Clinical Compound Library Plus;Bioactive Compound Library Plus;Apoptosis Compound Library;Cell […]
For research use only. We do not sell to patients. Dilevalol-d3 hydrochloride CAS No. : 2734920-41-1 Biological Activity：Dilevalol-d3 hydrochloride is the deuterium labeled Dilevalol hydrochloride. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent […]