Tag: Inhibitor|Agonist

For research use only. We do not sell to patients. Guanabenz hydrochloride CAS No. : 23113-43-1 Biological Activity：Guanabenz hydrochloride is an orally active α-2-adrenoceptor agonist. Guanabenz hydrochloride has antihypertensive effect and antiparasitic activity. Guanabenz hydrochloride interferes ER stress-signalling and has protective effects in cardiac myocytes. Guanabenz hydrochloride also is used for the research of high […]

For research use only. We do not sell to patients. Leelamine CAS No. : 1446-61-3 Biological Activity：Leelamine is a weak agonist of cannabinoid receptors CB1 and CB2. Leelamine also inhibits pyruvate dehydrogenase kinases (PDKs). Leelamine exhibits anti-tumor activity. Research Area：Cancer Targets：PDHK|Cannabinoid Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Kinase Inhibitor Library;Metabolism/Protease Compound Library;Neuronal […]

For research use only. We do not sell to patients. Loteprednol Etabonate-d3 Biological Activity：Loteprednol Etabonate-d3 is the deuterium labeled Loteprednol Etabonate. Loteprednol etabonate (LE) is an orally active “soft” steroid belonging to a unique class of glucocorticoids. Loteprednol etabonate (LE) exhibits anti-inflammatory activity and has been used in optometry and ophthalmology[2][3]. Research Area：Infection|Endocrinology|Inflammation/Immunology Targets：Glucocorticoid Receptor|Bacterial|Antibiotic […]

For research use only. We do not sell to patients. WAY-100635 Maleate CAS No. : 1092679-51-0 Biological Activity：WAY-100635 maleate is a potent and selective 5-hydroxytryptamine 1A (5-HT1A) receptor antagonist with an IC50 value of 0.91 nM and Ki value of 0.39 nM. WAY-100635 maleate has pIC50 values for 5-HT1A and α1-adrenergic receptors of 8.9 and […]

For research use only. We do not sell to patients. (Z)-Capsaicin-d3 Biological Activity：(Z)-Capsaicin-d3 (Zucapsaicin-d3) is the deuterium labeled (Z)-Capsaicin. (Z)-Capsaicin is the cis isomer of capsaicin, acts as an orally active TRPV1 agonist, and is used in the research of neuropathic pain[2]. Research Area：Neurological Disease Targets：HSV|TRP Channel Related Small Molecules:V116517;Isoborneol;GSK2332255B;Pregnenolone monosulfate sodium;Vidarabine monohydrate;TRPC5-IN-4;OptoBI-1;SB-705498;TRPC3/6-IN-1;ABT-239;Pyr3;Asivatrep;Ononetin;TRPM8 antagonist 3;FEMA […]

For research use only. We do not sell to patients. Camphor-d6 Biological Activity：Camphor-d6 ((±)-Camphor-d6) is the deuterium labeled Camphor. Camphor ((±)-Camphor) is a topical anti-infective and anti-pruritic and internally as a stimulant and carminative. However, Camphor is poisonous when ingested. Antiviral, antitussive, and anticancer activities. Camphor is a TRPV3 agonist[2]. Research Area：Cancer|Infection|Inflammation/Immunology Targets：Influenza Virus|TRP Channel […]

For research use only. We do not sell to patients. CAY10590 CAS No. : 1101136-50-8 Biological Activity：CAY10590 (GK115) is an inhibitor of secreted phospholipase A2 (sPLA2) and can be used for the research of chronic inflammatory kidney diseases. Research Area：Inflammation/Immunology Targets：Prostaglandin Receptor|Phospholipase Related Small Molecules:GK563;DPTIP;Cambinol;Neomycin sulfate;ONO-RS-082;Omidenepag isopropyl;DG-041;8-Isoprostaglandin E2;BAY-6672;trans-Isoferulic acid;ARN19874;GSK-269984A;KMN-80;LEI-401;ST271;SC 51089;Melittin TFA;(S)-Bromoenol lactone;p-Hydroxycinnamic acid;GK187;D-Erythro-dihydrosphingosine-d7;Pexopiprant;FKGK11;Dinoprost;PACOCF3 Trending products：Recombinant […]

For research use only. We do not sell to patients. L-Glutamine-1-13C CAS No. : 159663-16-8 Biological Activity：L-Glutamine-1-13C (L-Glutamic acid 5-amide-1-13C) is the 13C-labeled L-Glutamine. L-Glutamine (L-Glutamic acid 5-amide) is a non-essential amino acid present abundantly throughout the body and involved in many metabolic processes. L-Glutamine provides a source of carbons for oxidation in some cells[2]. […]

For research use only. We do not sell to patients. L-Glutamine-15N-1 CAS No. : 59681-32-2 Biological Activity：L-Glutamine-15N-1 (L-Glutamic acid 5-amide-15N-1) is the 15N-labeled L-Glutamine. L-Glutamine (L-Glutamic acid 5-amide) is a non-essential amino acid present abundantly throughout the body and involved in many metabolic processes. L-Glutamine provides a source of carbons for oxidation in some cells[2]. […]

For research use only. We do not sell to patients. Selgantolimod CAS No. : 2004677-13-6 Biological Activity：Selgantolimod (GS-9688) is an orally active, potent and selective toll-like receptor 8 (TLR8) agonist for the treatment of hepatitis B virus (HBV) and human immunodeficiency virus (HIV) infection[2][3]. Research Area：Infection Targets：HBV|Toll-like Receptor (TLR) Related Screening Libraries:Drug Repurposing Compound Library […]