Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. EZH2-IN-2 CAS No. : 2238821-31-1 Biological Activity：EZH2-IN-2 is a EZH2 inhibitor extracted from patent WO2018133795A1, Compound Example 69, with an IC50 of 64 nM. EZH2-IN-2 can be used for the research of cancer or precancerous condition related to EZH2 activity. Research Area：Cancer Targets：Histone Methyltransferase Related […]
For research use only. We do not sell to patients. Bromoacetamido-PEG8-Boc CAS No. : 2055041-16-0 Biological Activity：Bromoacetamido-PEG8-Boc is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs. Research Area：Cancer Targets：PROTAC Linkers Related Small Molecules:N-(Mal-PEG6)-N-bis(PEG7-TCO);Propargyl-PEG2-CH2COOH;NHS ester-PEG10-COOH;Tos-PEG5-Boc;Bis-PEG6-NHS ester;Azide-PEG12-alcohol;Fmoc-PEG6-NHS ester;Boc-C1-PEG3-C4-OBn;Boc-NH-PEG8-C2-Br;Propargyl-PEG14-Boc;m-PEG21-OH;Bromo-PEG3-THP;m-PEG8-Ms;Bis-PEG10-NHS ester;TCO-PEG3-acid;m-PEG8-DBCO;Azide-PEG6-Tos;Acid-PEG3-C2-Boc;m-PEG-mal (MW 2000);Benzyl-PEG7-t-butyl ester;Boc-Pip-alkyne-Ph-COOH;Biotin-PEG2-C6-azide;Bis-PEG4-acid;Active-mono-sulfone-PEG8-acid;Br-PEG6-C2-NHBoc;HO-PEG8-CH2COOH;NH2-PEG4-CH2CH2COOH;N-(Propargyl-PEG2)-N-Boc-PEG3-t-butyl ester;Carboxy-PEG2-sulfonic acid Trending products：Recombinant Proteins | Bioactive Screening Libraries | […]
For research use only. We do not sell to patients. Antitubercular agent-28 CAS No. : 2460651-10-7 Biological Activity：Antitubercular agent-28 (compound 2) is a potent antitubercular agent with an IC50 value of 1.5 µM, an MIC value of 4.5 µM, an IC90 value of 2.5 µM. Antitubercular agent-28 shows antimycobacterial activity for resistant isolates of Mycobacterium […]
For research use only. We do not sell to patients. Myelin Basic Protein CAS No. : 126768-94-3 Biological Activity：Myelin Basic Protein (MHP4-14), a synthetic peptide comprising residues 4-14 of myelin basic protein, is a very selective PKC substrate (Km=7 μM). Myelin Basic Protein is not phosphorylated by cyclic AMP-dependent protein kinase, casein kinases I and […]
For research use only. We do not sell to patients. Tenofovir-C3-O-C15-CF3 ammonium CAS No. : 2611373-80-7 Biological Activity：Tenofovir-C3-O-C15-CF3 (ammonium) exhibits substantially longer t1/2 values than tenofovir in human liver microsomes, potent anti-HIV activity in vitro, and enhances pharmacokinetic properties in vivo. Research Area：Infection Targets：HIV Related Small Molecules:HIV-1 TAT (48-60);Seletracetam lithium;HIV-IN-2;Triptonine B;FC131;Peritassine A;Flavopiridol;TAT (48-57);FGI-106 tetrahydrochloride;(Z)-9-Propenyladenine;Apabetalone;Decanoyl-RVKR-CMK TFA;ONX-0914 […]
For research use only. We do not sell to patients. Magnesium citrate CAS No. : 3344-18-1 Biological Activity：Magnesium citrate is a magnesium salt form that provides efficient penetration into brain and muscle tissue. Magnesium citrate increases pain threshold and reduces TLR4 concentration in the brain. Orally active. Research Area：Neurological Disease Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 […]
For research use only. We do not sell to patients. TC-S 7009 CAS No. : 1422955-31-4 Biological Activity：TC-S 7009 is a potent and selective HIF-2α inhibitor with a Kd of 81 nM. TC-S 7009 is more selective for HIF-2α than HIF-1α (Kd ≫ 5 μM). TC-S 7009 disrupts HIF-2α heterodimerization, decreases DNA-binding activity, and reduces […]
For research use only. We do not sell to patients. BMS-690514 CAS No. : 859853-30-8 Biological Activity：BMS-690514 is a potent and orally active inhibitor of EGFR and VEGFR; has IC50s of 5, 20 and 60 nM for EGFR, HER 2 and HER 4, respectively. Research Area：Cardiovascular Disease|Cancer Targets：EGFR|VEGFR Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical […]
For research use only. We do not sell to patients. Fmoc-L-photo-methionine CAS No. : 945859-89-2 Biological Activity：Fmoc-L-photo-methionine is a Methionine (HY-13694) derivative. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC […]
For research use only. We do not sell to patients. Ochromycinone CAS No. : 111540-00-2 Biological Activity：Ochromycinone ((Rac)-STA-21) is a natural antibiotic and a STAT3 inhibitor. Ochromycinone can inhibits STAT3 DNA binding activity, STAT3 dimerization. Ochromycinone has anticancer and antimicrobial activity[2]. Research Area：Cancer|Infection Targets：STAT|Bacterial Related Screening Libraries:Natural Product Library Plus;Bioactive Compound Library Plus;Anti-Infection Compound Library;Immunology/Inflammation […]