2023 - epigenetics modulation frontier

PKI 14-22 amide,myristoylated TFA

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. PKI 14-22 amide,myristoylated TFA Biological Activity：PKI 14-22 amide,myristoylated TFA is a potent cAMP-dependent PKA inhibitor. PKI 14-22 amide,myristoylated TFA reduces the IgG-mediated phagocytic response and also inhibits neutrophil adhesion. Research Area：Cancer Targets：PKA Related Screening Libraries:Bioactive Compound Library Plus;Peptide Library; Related Small Molecules:Staurosporine;Malantide;DS89002333;Rp-8-CPT-cAMPS sodium;PF-4950834;Warangalone;STAD 2;AT13148;CCG215022;KT5720;8-Bromo-cAMP sodium […]

Acid-PEG3-C2-Boc

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Acid-PEG3-C2-Boc CAS No. : 1807539-06-5 Biological Activity：Acid-PEG3-C2-Boc is a PEG- and Alkyl/ether-based PROTAC linker can be used in the synthesis of PROTACs for the degradation of EGFR and inhibition of mTOR[2]. Research Area：Cancer Targets：PROTAC Linkers Related Small Molecules:N-(Mal-PEG6)-N-bis(PEG7-TCO);Propargyl-PEG2-CH2COOH;NHS ester-PEG10-COOH;Tos-PEG5-Boc;Bis-PEG6-NHS ester;Azide-PEG12-alcohol;Fmoc-PEG6-NHS ester;Boc-C1-PEG3-C4-OBn;Boc-NH-PEG8-C2-Br;Propargyl-PEG14-Boc;m-PEG21-OH;Bromo-PEG3-THP;m-PEG8-Ms;Bis-PEG10-NHS ester;TCO-PEG3-acid;m-PEG8-DBCO;Azide-PEG6-Tos;m-PEG-mal (MW 2000);Benzyl-PEG7-t-butyl ester;Boc-Pip-alkyne-Ph-COOH;Biotin-PEG2-C6-azide;Bis-PEG4-acid;Active-mono-sulfone-PEG8-acid;Br-PEG6-C2-NHBoc;HO-PEG8-CH2COOH;NH2-PEG4-CH2CH2COOH;N-(Propargyl-PEG2)-N-Boc-PEG3-t-butyl […]

Ibrutinib dimer

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Ibrutinib dimer CAS No. : 2031255-23-7 Biological Activity：Ibrutinib dimer is a Dimer of Ibrutinib. Ibrutinib dimer is an impurity of Ibrutinib. Ibrutinib is a selective, irreversible Btk inhibitor with an IC50 of 0.5 nM[2]. Research Area：Cancer Targets：Btk Related Small Molecules:JAK3/BTK-IN-1;Elsubrutinib;ARQ 531;PF-06250112;PCI 29732;CHMFL-EGFR-202;Avitinib;RN486;GDC-0834 Racemate;Spebrutinib besylate;Vecabrutinib;BMX-IN-1;Tolebrutinib;BTK-IN-16;(R)-Zanubrutinib;Pirtobrutinib;CTA056;EGFR-IN-40;QL-X-138;ACP-5862;BTK-IN-12;JAK3/BTK-IN-4;JAK3/BTK-IN-6;BTK inhibitor […]

Lenampicillin hydrochloride

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Lenampicillin hydrochloride CAS No. : 80734-02-7 Biological Activity：Lenampicillin hydrochloride (KBT 1585 hydrochloride) is an orally active prodrug of Ampicillin and is an effective beta-lactam antibacterial agent that inhibits bacterial penicillin-binding proteins (transpeptidase). Lenampicillin hydrochloride has improved absorption and decreased side effects compares to Ampicillin and […]

Pregnenolone monosulfate sodium

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Pregnenolone monosulfate sodium CAS No. : 1852-38-6 Biological Activity：Pregnenolone monosulfate sodium (3β-Hydroxy-5-pregnen-20-one monosulfate sodium) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate sodium acts as a signaling-specific inhibitor of cannabinoid CB1 receptor, inhibits the effects of tetrahydrocannabinol […]

His-Pro

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. His-Pro CAS No. : 20930-58-9 Biological Activity：His-Pro is a dipeptide consisting of histidyl and proline. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent […]

Notoginsenoside Fc

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Notoginsenoside Fc CAS No. : 88122-52-5 Biological Activity：Notoginsenoside Fc, a protopanaxadiol- (PPD-) type saponin isolated from the leaves of Panax notoginseng, effectively counteracts platelet aggregation. Notoginsenoside Fc can accelerate reendothelialization following vascular injury in diabetic rats by promoting autophagy. Research Area：Cardiovascular Disease Targets：Autophagy Related Screening […]

Lu AE98134

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Lu AE98134 CAS No. : 849000-18-6 Biological Activity：Lu AE98134, an activator of voltage-gated sodium channels, acts as a partly selective Nav1.1 channels positive modulator. Lu AE98134 also increases the activity of Nav1.2 and Nav1.5 channels but not of Nav1.4, Nav1.6 and Nav1.7 channels. Lu AE98134 […]

Antibacterial agent 45

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. Antibacterial agent 45 CAS No. : 1426572-50-0 Biological Activity：Antibacterial agent 45, an antibacterial agent, significantly lowers MIC value of antibacterial agent Ceftazidime. Research Area：Infection Targets：Bacterial Related Small Molecules:Sandramycin;LLO (91-99);Gepotidacin;Oritavancin;Azlocillin sodium salt;Herbimycin A;Leucomycin;Isouvaretin;Antibacterial agent 99;Nafcillin;Antitubercular agent-28;Ochromycinone;Staurosporine;Nucleocidin;(±)-Leucine-13C-1;Ciclopirox-d11;Ciclopirox olamine;Clotrimazole-d5;SQ109;Neomycin sulfate;Bauer-7-ene-3β,16α-diol;Aminothiazole Trending products：Recombinant Proteins | Bioactive Screening Libraries | […]

ATX inhibitor 22

Posted on January 16, 2023 by haoyuan2014

For research use only. We do not sell to patients. ATX inhibitor 22 Biological Activity：ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) with IC50 of 218 nM but lost its inhibitory activity of LPAR1. Research Area：Cancer Targets：Phosphodiesterase (PDE) Related Small Molecules:Senazodan hydrochloride;(E/Z)-HA155;Enpp/Carbonic anhydrase-IN-1;Carbazeran citrate;Bay 60-7550;BC11-38;Deltarasin hydrochloride;Glaucine;Ziritaxestat;Udenafil-d7;D159687;ITI-214;PDE10-IN-5;ICI 153110;Furamidine dihydrochloride;ML-030;PDE4-IN-10;Mirodenafil-d7 dihydrochloride;PDE1-IN-4;PDE4B-IN-3;Cirsimarin;PF-03049423;IBMX;Pimobendan;Gisadenafil besylate;S32826 disodium Trending products：Recombinant […]