Tag: Inducer|Inhibitor

For research use only. We do not sell to patients. JKE-1674 CAS No. : 2421119-60-8 Biological Activity：JKE-1674 is an orally active glutathione peroxidase 4 (GPX4) inhibitor and an active metabolite of GPX4 inhibitor ML-210. JKE-1674, an analog of ML-210 in which the nitroisoxazole ring is replaced with an α-nitroketoxime. JKE-1674 can convert into a nitrile […]

For research use only. We do not sell to patients. IST5-002 CAS No. : 13484-66-7 Biological Activity：IST5-002, a potent Stat5a/b inhibitor, selectively inhibits transcriptional activity of Stat5a/b (IC50s: 1.5 μM for Stat5a, 3.5 μM for Stat5b). IST5-002 inducs cell apoptotic and death of prostate cancer cells and chronic myeloid leukemia (CML) cells. IST5-002 can be […]

For research use only. We do not sell to patients. Quinidine sulfate dihydrate CAS No. : 6591-63-5 Biological Activity：Quinidine sulfate dihydrate is an antiarrhythmic agent. Quinidine sulfate dihydrate is a potent, orally active, selective cytochrome P450db inhibitor. Quinidine sulfate dihydrate is also a K+ channel blocker with an IC50 of 19.9 μM, and can induce […]

For research use only. We do not sell to patients. IU1 CAS No. : 314245-33-5 Biological Activity：IU1 is a special Usp14 inhibitor with an IC50 of 4-5 μM. Research Area：Cardiovascular Disease Targets：Autophagy|Deubiquitinase Related Screening Libraries:Bioactive Compound Library Plus;Cell Cycle/DNA Damage Compound Library;Autophagy Compound Library;Peptidomimetic Library;Anti-Aging Compound Library;Anti-Cardiovascular Disease Compound Library;Ubiquitination Compound Library;Targeted Diversity Library; Related […]

For research use only. We do not sell to patients. Aloperine CAS No. : 56293-29-9 Biological Activity：Aloperine is an alkaloid in sophora plants such as Sophora alopecuroides L, which has shown anti-cancer, anti-inflammatory and anti-virus properties. Aloperine is widely used to treat patients with allergic contact dermatitis eczema and other skin inflammation in China[2]. Aloperine […]

For research use only. We do not sell to patients. Multi-kinase-IN-1 CAS No. : 2470807-67-9 Biological Activity：Multi-kinase-IN-1 (Compound 11k) is a potent kinase inhibitor with antitumor activity. Multi-kinase-IN-1 induces cell apoptosis, and can be studied for colorectal cancer. Research Area：Cancer Targets：c-Met/HGFR|Src|Apoptosis|PDGFR|TAM Receptor Related Small Molecules:Physalin A;Bomedemstat ditosylate;Enpp/Carbonic anhydrase-IN-1;GK563;Calpeptin;Lobetyolin;KB SRC 4;Tirbanibulin dihydrochloride;AMG-208;D6808;BJE6-106;Dinaciclib;Ecteinascidin 770;MDM2-p53-IN-15;AT9283;Staurosporine;SNS-032;C188-9;ZLDI-8;Topoisomerase I/II inhibitor 3;Xevinapant;Mangiferin;Cambinol;Antioxidant […]

For research use only. We do not sell to patients. Oxyresveratrol CAS No. : 29700-22-9 Biological Activity：Oxyresveratrol (trans-Oxyresveratrol) is a potent naturally occurring antioxidant and free radical scavenger (IC50 of 28.9 µM against DPPH free radicals). Oxyresveratrol is potent and noncompetitive tyrosinase inhibitor with an IC50 value of 1.2 µM for mushroom tyrosinase. Oxyresveratrol is […]

For research use only. We do not sell to patients. STF-118804 CAS No. : 894187-61-2 Biological Activity：STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50

For research use only. We do not sell to patients. L-threo-Sphingosine CAS No. : 25695-95-8 Biological Activity：L-threo-Sphingosine is a potent MAPK inhibitor. L-threo-Sphingosine induces apoptosis and clear DNA fragmentation. L-threo-Sphingosine shows anticancer effect. Research Area：Cancer Targets：p38 MAPK|Apoptosis Related Small Molecules:Physalin A;Bomedemstat ditosylate;Enpp/Carbonic anhydrase-IN-1;GK563;Calpeptin;Lobetyolin;BJE6-106;Dinaciclib;Ecteinascidin 770;MDM2-p53-IN-15;AT9283;Staurosporine;SNS-032;C188-9;ZLDI-8;Topoisomerase I/II inhibitor 3;Xevinapant;Mangiferin;Cambinol;Antioxidant agent-5;Apoptosis inducer 9;Bafetinib;Cyclovirobuxine D;STAT3-IN-10;Rigosertib sodium Trending products：Recombinant Proteins  […]

For research use only. We do not sell to patients. Arctigenin CAS No. : 7770-78-7 Biological Activity：Arctigenin ((-)-Arctigenin), a biologically active lignan, can be used as an antitumor agent. Arctigenin exhibits potent antioxidant, anti-inflammatory and antiviral (influenza A virus) activities. Arctigenin can be used for the research of metabolic disorders, and central nervous system dysfunctions[2][3]. […]