Tag: Antagonist|Agonist

For research use only. We do not sell to patients. Urapidil D6 Biological Activity：Urapidil D6 is a deuterium labeled Urapidil. Urapidil is an α1-adrenoreceptor antagonist and a 5-HT1A receptor agonist. Research Area：Endocrinology|Neurological Disease Targets：Adrenergic Receptor|5-HT Receptor Related Small Molecules:F 13714;Mosapride-d5;Todralazine;ARC 239 dihydrochloride;Nuciferine;Yohimbine;Glaucine;Salbutamol;Renzapride;BI-167107;LY 344864 racemate;Harmine hydrochloride;Talibegron hydrochloride;Valerenic acid;Arotinolol;SR59230A;Melitracen-d6 hydrochloride;WAY-100635 Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  […]

For research use only. We do not sell to patients. Cinitapride CAS No. : 66564-14-5 Biological Activity：Cinitapride is an orally active 5-HT4 agonist and D2 antagonist. Cinitapride shows gastroprotective properties on mucosal injury. Cinitapride can be used in functional dyspepsia (FD) and gastroesophageal reflux disease (GERD) research[2][3]. Research Area：Metabolic Disease Targets：Dopamine Receptor|Histamine Receptor Related Small […]

For research use only. We do not sell to patients. Candesartan CAS No. : 139481-59-7 Biological Activity：Candesartan (CV 11974) is an orally active angiotensin II AT1-Receptor blocker and PPAR-γ agonist. Candesartan has potent and long-lasting antihypertensive effects. Candesartan can be used for the research of hypertension, chronic heart failure (CHF) and Traumatic brain injury (TBI)[2][3]. […]

For research use only. We do not sell to patients. Urapidil-d4 hydrochloride CAS No. : 1794979-63-7 Biological Activity：Urapidil-d4 hydrochloride is the deuterium labeled Urapidil hydrochloride. Urapidil hydrochloride is an α1-adrenoceptor antagonist and 5-HT1A receptor agonist[2]. Research Area：Cardiovascular Disease|Endocrinology Targets：Adrenergic Receptor|5-HT Receptor Related Small Molecules:F 13714;Mosapride-d5;Todralazine;ARC 239 dihydrochloride;Nuciferine;Yohimbine;Glaucine;Salbutamol;Renzapride;BI-167107;LY 344864 racemate;Harmine hydrochloride;Talibegron hydrochloride;Valerenic acid;Arotinolol;SR59230A;Melitracen-d6 hydrochloride;WAY-100635 Trending products：Recombinant […]

For research use only. We do not sell to patients. Clozapine N-oxide CAS No. : 34233-69-7 Biological Activity：Clozapine N-oxide is a major metabolite of Clozapine and a human muscarinic designer receptors (DREADDs) agonist. Clozapine N-oxide activates the DREADD receptor hM3Dq and hM4Di. Clozapine N-oxide can cross the blood-brain barrier[2][3][4]. Clozapine is a potent dopamine antagonist […]

For research use only. We do not sell to patients. GTS-21 dihydrochloride CAS No. : 156223-05-1 Biological Activity：GTS-21 dihydrochloride is a selective alpha7 nicotinic acetylcholine receptor (α7-nAChR) agonist with anti‑inflammatory and cognition‑enhancing activities. GTS-21 dihydrochloride is also a α4β2 (Ki=20 nM for humanα4β2) and 5-HT3A receptor (IC50=3.1 μM) antagonist[2]. Research Area：Inflammation/Immunology Targets：nAChR|5-HT Receptor Related Screening […]

For research use only. We do not sell to patients. 4-PPBP maleate CAS No. : 201216-39-9 Biological Activity：4-PPBP maleate is a potent σ 1 receptor ligand and agonist. 4-PPBP maleate is a non-competitive, selective NR1a/2B NMDA receptors (expressed in Xenopus oocytes) antagonist. 4-PPBP maleate provides neuroprotection[2][3]. Research Area：Neurological Disease Targets：Sigma Receptor|iGluR Related Small Molecules:CIQ;Quinolinic acid-d3;1-Aminocyclobutanecarboxylic […]

For research use only. We do not sell to patients. Urapidil-d3 CAS No. : 1398066-08-4 Biological Activity：Urapidil-d3 is the deuterium labeled Urapidil. Urapidil is an α1 adrenoreceptor antagonist and a 5-HT1A receptor agonist. Research Area：Neurological Disease|Endocrinology Targets：Adrenergic Receptor|5-HT Receptor Related Small Molecules:F 13714;Mosapride-d5;Todralazine;ARC 239 dihydrochloride;Nuciferine;Yohimbine;Glaucine;Salbutamol;Renzapride;BI-167107;LY 344864 racemate;Harmine hydrochloride;Talibegron hydrochloride;Valerenic acid;Arotinolol;SR59230A;Melitracen-d6 hydrochloride;WAY-100635 Trending products：Recombinant Proteins  |  […]

For research use only. We do not sell to patients. Quetiapine-d8 hemifumarate Biological Activity：Quetiapine-d8 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a 5-HT receptors agonist with a pEC50 of 4.77 for human 5-HT1A receptor. Quetiapine hemifumarate is a dopamine receptor antagonist with a pIC50 of 6.33 for human D2 receptor. Quetiapine hemifumarate […]

For research use only. We do not sell to patients. Ursodeoxycholic acid sodium CAS No. : 2898-95-5 Biological Activity：Ursodeoxycholic acid (Ursodeoxycholate) sodium is a secondary bile acid issued from the transformation of (cheno)deoxycholic acid by intestinal bacteria, acting as a key regulator of the intestinal barrier integrity and essential for lipid metabolism. Ursodeoxycholic acid sodium […]