Tag: Antagonist

For research use only. We do not sell to patients. Ecastolol CAS No. : 77695-52-4 Biological Activity：Ecastolol is a beta adrenergic receptor antagonist, with antianginal activities. Research Area：Cardiovascular Disease|Endocrinology Targets：Adrenergic Receptor Related Small Molecules:Todralazine;ARC 239 dihydrochloride;Yohimbine;Glaucine;Salbutamol;BI-167107;Talibegron hydrochloride;Arotinolol;SR59230A;Higenamine hydrochloride;Navafenterol saccharinate;Isoprenaline hydrochloride;Bevantolol;Zilpaterol-d7;Ritanserin;A55453;Povafonidine;β3-AR agonist 1;Tulobuterol;AGN 192836;KUC-7322;Oxyfedrine;Urapidil hydrochloride;Detomidine hydrochloride;Oxprenolol-d7 hydrochloride;Nicergoline;Synephrine hemitartrate;ADRA1D receptor antagonist 1;Solabegron Trending products：Recombinant Proteins  |  Bioactive […]

For research use only. We do not sell to patients. OPC-28326 CAS No. : 167626-17-7 Biological Activity：OPC-28326 is a selective peripheral vasodilator and an angatonist of α2-adrenergic receptor, with Ki of 2040, 285, and 55 nM for α2A-, α2B- and α2C-adrenoceptors, respectively. Research Area：Cardiovascular Disease|Endocrinology Targets：Adrenergic Receptor Related Small Molecules:Todralazine;ARC 239 dihydrochloride;Yohimbine;Glaucine;Salbutamol;BI-167107;Talibegron hydrochloride;Arotinolol;SR59230A;Higenamine hydrochloride;Navafenterol saccharinate;Isoprenaline hydrochloride;Bevantolol;Zilpaterol-d7;Ritanserin;A55453;Povafonidine;β3-AR […]

For research use only. We do not sell to patients. PD-159020 CAS No. : 177904-00-6 Biological Activity：PD-159020 is a non-selective ETA/ETB antagonist, with IC50s of 30 and 50 nM for hETA and hETB, respectively. Research Area：Cardiovascular Disease|Endocrinology Targets：Endothelin Receptor Related Small Molecules:BQ-788;[Asn18] Endothelin-1, human;Endothelin-3, human, mouse, rabbit, rat TFA;IRL 2500;Sarafotoxin S6c;Sarafotoxin S6a;ANP (1-30), frog;IRL-1620 TFA;Tezosentan;ACT-373898;Ro […]

For research use only. We do not sell to patients. Elisartan CAS No. : 149968-26-3 Biological Activity：Elisartan is an orally active non-peptide pro-drug of angiotensin II AT1 receptor antagonist HN-12206, and shows anti-hypertension activities. Research Area：Cardiovascular Disease|Endocrinology Targets：Angiotensin Receptor Related Small Molecules:Saralasin;A81988;EMD 66684;TD-0212;Angiotensin I/II (1-6) (TFA);YS-49;TRV055;TRV056;H-Val-Pro-Pro-OH TFA;Tranilast sodium;Angiotensin amide;L162389;L-159282;CGP48369;Pratosartan;TRV-120027 TFA;SL910102 Trending products：Recombinant Proteins  |  Bioactive […]

For research use only. We do not sell to patients. CP 316311 CAS No. : 175139-41-0 Biological Activity：CP 316311 is a potent and selective CRF1 receptor antagonist with an IC50 value of 6.8 nM. Research Area：Neurological Disease|Endocrinology Targets：CRFR Related Small Molecules:Stresscopin-related peptide (human);Sauvagine;CRF(6-33)(human) TFA;NBI-27914;Urocortin III, mouse;Emicerfont;R121919;Pexacerfont;Urotensin I TFA;Urocortin, rat TFA;Urocortin II, human TFA;α-Helical CRF(9-41);CP 376395;Urocortin, […]

For research use only. We do not sell to patients. LAS101057 CAS No. : 925676-48-8 Biological Activity：LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist. Research Area：Inflammation/Immunology Targets：Adenosine Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Immunology/Inflammation Compound Library;Small Molecule Immuno-Oncology Compound Library;Neurotransmitter Receptor Compound Library;Anti-Parkinson’s Disease Compound Library;Neurodegenerative Disease-related Compound Library; […]

For research use only. We do not sell to patients. RPR104632 CAS No. : 154106-92-0 Biological Activity：RPR104632 is a specific antagonist of NMDA receptor, with potent neuroprotective properties. Research Area：Neurological Disease Targets：iGluR Related Small Molecules:CIQ;Quinolinic acid-d3;1-Aminocyclobutanecarboxylic acid;Glycine-1-13C,15N;ZL006;PYD-106;NMDA-IN-2;JAMI1001A;(S)-Willardiine;Fanapanel;(S)-AMPA;L-Glutamic acid-15N,d5;PDZ1 Domain inhibitor peptide TFA;Ifenprodil tartrate;Rislenemdaz;Coluracetam;Flupirtine-d4 hydrochloride;DL-Phenylalanine-d5 hydrochloride;NMDA;CFM-2;Lanicemine dihydrochloride;L-Phenylalanine-13C9;VSGLNPSLWSIFGLQFILLWLVSGSRHYLW TFA;L-Glutamic acid monosodium salt;Glycine-15N;Ibotenic acid;GYKI-47261 dihydrochloride;Sunifiram Trending products：Recombinant Proteins  […]

For research use only. We do not sell to patients. Pamatolol CAS No. : 59110-35-9 Biological Activity：Pamatolol is a cardioselective beta-adrenoceptor antagonist without sympathomimetic activity. Research Area：Cardiovascular Disease|Endocrinology Targets：Adrenergic Receptor Related Small Molecules:Todralazine;ARC 239 dihydrochloride;Yohimbine;Glaucine;Salbutamol;BI-167107;Talibegron hydrochloride;Arotinolol;SR59230A;Higenamine hydrochloride;Navafenterol saccharinate;Isoprenaline hydrochloride;Bevantolol;Zilpaterol-d7;Ritanserin;A55453;Povafonidine;β3-AR agonist 1;Tulobuterol;AGN 192836;KUC-7322;Oxyfedrine;Urapidil hydrochloride;Detomidine hydrochloride;Oxprenolol-d7 hydrochloride;Nicergoline;Synephrine hemitartrate;ADRA1D receptor antagonist 1;Solabegron Trending products：Recombinant Proteins  |  Bioactive Screening […]

For research use only. We do not sell to patients. MRZ 2-514 CAS No. : 202808-11-5 Biological Activity：MRZ 2-514 is an antagonist of the strychnine-insensitive modulatory site of the NMDA receptor (glycineB), with Ki of 33 μM. Research Area：Neurological Disease Targets：iGluR Related Screening Libraries:Bioactive Compound Library Plus; Related Small Molecules:CIQ;Quinolinic acid-d3;1-Aminocyclobutanecarboxylic acid;Glycine-1-13C,15N;ZL006;PYD-106;NMDA-IN-2;JAMI1001A;(S)-Willardiine;Fanapanel;(S)-AMPA;L-Glutamic acid-15N,d5;PDZ1 Domain inhibitor […]

For research use only. We do not sell to patients. SUN 1334H CAS No. : 607736-84-5 Biological Activity：SUN 1334H is a potent, orally active, highly selective H1 receptor antagonist, with Ki of 9.7 nM. Research Area：Inflammation/Immunology|Endocrinology Targets：Histamine Receptor Related Small Molecules:Tripelennamine;Brompheniramine-d6 maleate;Samelisant;Chlorphenoxamine;H3 receptor-MO-1;Diphenhydramine;ABT-239;Ketotifen fumarate;Ranitidine;Cetirizine;Diphenylpyraline hydrochloride;Loratadine-d5;Phenyltoloxamine;Ritanserin;BMY-25271;FRG8701;Mecamylamine hydrochloride;Cimetidine sulfoxide;Brompheniramine maleate;Tecastemizole;Famotidine-13C,d3;Bromazine-d6 hydrochloride Trending products：Recombinant Proteins  |  Bioactive Screening […]