Anipamil

For research use only. We do not sell to patients. Anipamil CAS No. : 83200-10-6 Biological Activity:Anipamil is a long-acting calcium channel blocker, used for the treatment of cardiovascular disease. Research Area:Cardiovascular Disease Targets:Calcium Channel Related Small Molecules:Benidipine hydrochloride;CaV1.3 antagonist-1;14-Deoxyandrographolide;(Rac)-MEM 1003;Glaucine;Efonidipine hydrochloride monoethanolate;L-Ascorbic acid sodium salt;Brompheniramine-d6 maleate;MRS 1523;Nilvadipine;Lercanidipine;CP-060;Anipamil-d25 hydrochloride;ISX-9;ω-Conotoxin MVIIC;Catharanthine;Thapsigargin;Tetrandrine;Ginsenoside Rd;Manidipine dihydrochloride;ω-Agatoxin IVA;AE0047 Hydrochloride;PDE1-IN-4 Trending […]

Wy 49051

For research use only. We do not sell to patients. Wy 49051 CAS No. : 113418-56-7 Biological Activity:Wy 49051 is a potent, orally active H1 receptor antagonist, with IC50 of 44 nM. Research Area:Inflammation/Immunology|Endocrinology Targets:Histamine Receptor Related Small Molecules:Tripelennamine;Brompheniramine-d6 maleate;Samelisant;Chlorphenoxamine;H3 receptor-MO-1;Diphenhydramine;ABT-239;Ketotifen fumarate;Ranitidine;Cetirizine;Diphenylpyraline hydrochloride;Loratadine-d5;Phenyltoloxamine;Ritanserin;BMY-25271;FRG8701;Mecamylamine hydrochloride;Cimetidine sulfoxide;Brompheniramine maleate;Tecastemizole;Famotidine-13C,d3;Bromazine-d6 hydrochloride Trending products:Recombinant Proteins  |  Bioactive Screening Libraries  |  […]

CGP48369

For research use only. We do not sell to patients. CGP48369 CAS No. : 135689-23-5 Biological Activity:CGP48369 is a nonpeptidic angiotensin II receptor antagonist, used for anti-hypertensive research. Research Area:Cardiovascular Disease|Endocrinology Targets:Angiotensin Receptor Related Small Molecules:Saralasin;A81988;EMD 66684;TD-0212;Angiotensin I/II (1-6) (TFA);YS-49;TRV055;TRV056;H-Val-Pro-Pro-OH TFA;Tranilast sodium;Angiotensin amide;L162389;L-159282;Elisartan;Pratosartan;TRV-120027 TFA;SL910102 Trending products:Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  […]

NRC-2694

For research use only. We do not sell to patients. NRC-2694 CAS No. : 936446-61-6 Biological Activity:NRC-2694 is an epidermal growth factor receptor (EGFR) antagonist with anti-cancer and anti-proliferative properties. Research Area:Cancer Targets:EGFR Related Screening Libraries:Covalent Screening Library Plus;Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;Immunology/Inflammation Compound Library;JAK/STAT Compound Library;Kinase Inhibitor Library;Protein […]

Elucaine

For research use only. We do not sell to patients. Elucaine CAS No. : 25314-87-8 Biological Activity:Elucaine is a muscarinic acetylcholine receptor antagonist with anti-ulcerative activity. Research Area:Inflammation/Immunology Targets:mAChR Related Small Molecules:VU0357017 hydrochloride;TBPB;Imidafenacin;Sabcomeline;MK-6884;Brompheniramine-d6 maleate;Navafenterol saccharinate;DREADD agonist 21;Cyclobuxine D;Brompheniramine maleate;Dexetimide;Anisodamine hydrobromide;Anisotropine bromide;PD 102807;Nebracetam hydrochloride;Muscarine-d9 iodide;Mazaticol;VU0455691;Arborine;Oxitropium Bromide;Propiverine hydrochloride;VU0152099;MHP 133;YM-58790;Rispenzepine;Phenglutarimid;Rapacuronium bromide;Ambutonium bromide;Temiverine hydrochloride;Procyclidine;M4 mAChR agonist-1;Camylofine Trending products:Recombinant Proteins  […]

Aligeron

For research use only. We do not sell to patients. Aligeron CAS No. : 70713-45-0 Biological Activity:Aligeron is a non-selective prostaglandin (PG) antagonist, and has vasodilatory properties. Research Area:Cardiovascular Disease|Endocrinology Targets:Prostaglandin Receptor Related Small Molecules:Omidenepag isopropyl;DG-041;8-Isoprostaglandin E2;BAY-6672;trans-Isoferulic acid;GSK-269984A;KMN-80;SC 51089;p-Hydroxycinnamic acid;Pexopiprant;Dinoprost;Sulprostone;Prostaglandin E2;CAY10471 Racemate;Fevipiprant;TG6-10-1;Cicaprost;ER-819762;MRE-269-d6;ONO-8130;KAG-308;KF 13218;Prostaglandin E2-d4 Trending products:Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  […]

SB-423562

For research use only. We do not sell to patients. SB-423562 CAS No. : 351490-27-2 Biological Activity:SB-423562 is a short-acting calcium-sensing receptor (CaR) antagonist. SB-423562 has the potential for osteoporosis research. Research Area:Inflammation/Immunology Targets:CaSR Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Immunology/Inflammation Compound Library;Protein-protein Interaction Inhibitor Library; Related Small Molecules:Calcium-Sensing Receptor Antagonists I;Calhex 231 […]

Org-10490

For research use only. We do not sell to patients. Org-10490 CAS No. : 83507-02-2 Biological Activity:Org-10490 is an antagonist of dopamine D1 receptor and dopamine D2 receptor, used for the treatment for psychiatric disease. Research Area:Neurological Disease Targets:Dopamine Receptor Related Small Molecules:Alizapride hydrochloride;Thioproperazine;Bromopride-d3;Nuciferine;Glaucine;SB-277011 dihydrochloride;MIF-1 TFA;Sulpiride;(Rac)-Razpipadon;Clebopride malate;WAY-100635;Flupentixol-d4 dihydrochloride;Cariprazine-d6 hydrochloride;Itopride-d6 hydrochloride;ONC206;Brexpiprazole S-oxide;cis-(Z)-Flupentixol dihydrochloride;D4R antagonist-1;U91356 Trending products:Recombinant […]

Terbogrel

For research use only. We do not sell to patients. Terbogrel CAS No. : 149979-74-8 Biological Activity:Terbogrel is an orally available thromboxane A2 receptor antagonist and a thromboxane A2 synthase inhibitor, with both IC50s of about 10 nM. Research Area:Cardiovascular Disease|Endocrinology Targets:Prostaglandin Receptor Related Small Molecules:Omidenepag isopropyl;DG-041;8-Isoprostaglandin E2;BAY-6672;trans-Isoferulic acid;GSK-269984A;KMN-80;SC 51089;p-Hydroxycinnamic acid;Pexopiprant;Dinoprost;Sulprostone;Prostaglandin E2;CAY10471 Racemate;Fevipiprant;TG6-10-1;Cicaprost;ER-819762;MRE-269-d6;ONO-8130;KAG-308;KF 13218;Prostaglandin E2-d4 […]

Rocastine

For research use only. We do not sell to patients. Rocastine CAS No. : 91833-49-7 Biological Activity:Rocastine is a selective, nonsedating H1 antagonist, acting as an antihistamine. Research Area:Inflammation/Immunology Targets:Histamine Receptor Related Small Molecules:Tripelennamine;Brompheniramine-d6 maleate;Samelisant;Chlorphenoxamine;H3 receptor-MO-1;Diphenhydramine;ABT-239;Ketotifen fumarate;Ranitidine;Cetirizine;Diphenylpyraline hydrochloride;Loratadine-d5;Phenyltoloxamine;Ritanserin;BMY-25271;FRG8701;Mecamylamine hydrochloride;Cimetidine sulfoxide;Brompheniramine maleate;Tecastemizole;Famotidine-13C,d3;Bromazine-d6 hydrochloride Trending products:Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  […]