Droperidol

For research use only. We do not sell to patients. Droperidol CAS No. : 548-73-2 Biological Activity:Droperidol is a Dopamine-2 Receptor Antagonist. Target: D2DR Droperidol is a butyrophenone, with anti-emetic, sedative and anti-anxiety properties. Research Area:Neurological Disease Targets:Dopamine Receptor Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;GPCR/G […]

RAGE antagonist peptide TFA

For research use only. We do not sell to patients. RAGE antagonist peptide TFA Biological Activity:RAGE antagonist peptide TFA is an advanced glycation end products (RAGE) antagonist. RAGE antagonist peptide TFA prevents RAGE from binding with several of its most important ligands, including HMGB-1, S100P, and S100A4. RAGE antagonist peptide TFA possesses anti-tumor and anti-inflammatory […]

L-Phenylalanine

For research use only. We do not sell to patients. L-Phenylalanine CAS No. : 63-91-2 Biological Activity:L-Phenylalanine ((S)-2-Amino-3-phenylpropionic acid) is an essential amino acid isolated from Escherichia coli. L-Phenylalanine is a α2δ subunit of voltage-dependent Ca+ channels antagonist with a Ki of 980 nM. L-phenylalanine is a competitive antagonist for the glycine- and glutamate-binding sites […]

[Des-His1,Glu9]-Glucagon amide TFA

For research use only. We do not sell to patients. [Des-His1,Glu9]-Glucagon amide TFA Biological Activity:[Des-His1,Glu9]-Glucagon amide TFA is a potent and peptide antagonist of the glucagon receptor, with a pA2 of 7.2. [Des-His1,Glu9]-Glucagon amide TFA is potentially useful in the study of the pathogenesis of diabetes. Research Area:Metabolic Disease Targets:GCGR Related Screening Libraries:Bioactive Compound Library […]

Diphenhydramine-d6 hydrochloride

For research use only. We do not sell to patients. Diphenhydramine-d6 hydrochloride CAS No. : 1189986-72-8 Biological Activity:Diphenhydramine-d6 hydrochloride is the deuterium labeled Diphenhydramine hydrochloride. Diphenhydramine hydrochloride is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine hydrochloride can across the ovine blood-brain barrier (BBB)[2]. Research Area:Inflammation/Immunology|Endocrinology Targets:Histamine Receptor|Endogenous Metabolite Related Small Molecules:D-α-Hydroxyglutaric acid disodium;Nicotinamide […]

Pranlukast hemihydrate

For research use only. We do not sell to patients. Pranlukast hemihydrate CAS No. : 150821-03-7 Biological Activity:Pranlukast hemihydrate is a highly potent, selective and competitive antagonist of peptide leukotrienes. Pranlukast inhibits [3H]LTE4, [3H]LTD4, and [3H]LTC4 bindings to lung membranes with Kis of 0.63±0.11, 0.99±0.19, and 5640±680 nM, respectively. Research Area:Inflammation/Immunology Targets:Leukotriene Receptor|Endogenous Metabolite Related […]

SBI-115

For research use only. We do not sell to patients. SBI-115 CAS No. : 882366-16-7 Biological Activity:SBI-115 is a TGR5 (GPCR19) antagonist. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5. Research Area:Others Targets:G protein-coupled Bile Acid Receptor 1 Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Anti-Obesity Compound Library;Lipid Metabolism Compound Library […]

Hydroxyzine pamoate

For research use only. We do not sell to patients. Hydroxyzine pamoate CAS No. : 10246-75-0 Biological Activity:Hydroxyzine pamoate is a histamine H1-receptor antagonist. Target: Histamine H1-Receptor Hydroxyzine inhibits carbachol (10 μM)-induced serotonin release by 34% at 10 μM, by 25% 1 μM and by 17% 0.1 μM in pretreated bladder slices for 60 min […]

[D-Phe2,D-Ala6]-LH-RH

For research use only. We do not sell to patients. [D-Phe2,D-Ala6]-LH-RH CAS No. : 54784-44-0 Biological Activity:[D-Phe2,D-Ala6]-LH-RH is a potent LH-RH antagonist. [D-Phe2,D-Ala6]-LH-RH shows anti-LH/FSH-RH and antiovulatory activities. Research Area:Endocrinology Targets:Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products:Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural […]

Rat CGRP-(8-37)

For research use only. We do not sell to patients. Rat CGRP-(8-37) CAS No. : 129121-73-9 Biological Activity:Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist. Research Area:Neurological Disease|Cardiovascular Disease Targets:CGRP Receptor Related Screening Libraries:Bioactive Compound Library Plus;Peptide Library; Related Small Molecules:Vazegepant hydrochloride;Adrenomedullin (16-31), human;MK-3207 Hydrochloride;α-CGRP, rat;Cagrilintide acetate;HTL22562;SUN B8155;Adrenomedullin (11-50), rat;Atogepant;β-CGRP, human TFA;Calcitonin (salmon);Calcitonin […]