Tag: Antagonist

For research use only. We do not sell to patients. Droperidol CAS No. : 548-73-2 Biological Activity：Droperidol is a Dopamine-2 Receptor Antagonist. Target: D2DR Droperidol is a butyrophenone, with anti-emetic, sedative and anti-anxiety properties. Research Area：Neurological Disease Targets：Dopamine Receptor Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;GPCR/G […]

For research use only. We do not sell to patients. RAGE antagonist peptide TFA Biological Activity：RAGE antagonist peptide TFA is an advanced glycation end products (RAGE) antagonist. RAGE antagonist peptide TFA prevents RAGE from binding with several of its most important ligands, including HMGB-1, S100P, and S100A4. RAGE antagonist peptide TFA possesses anti-tumor and anti-inflammatory […]

For research use only. We do not sell to patients. L-Phenylalanine CAS No. : 63-91-2 Biological Activity：L-Phenylalanine ((S)-2-Amino-3-phenylpropionic acid) is an essential amino acid isolated from Escherichia coli. L-Phenylalanine is a α2δ subunit of voltage-dependent Ca+ channels antagonist with a Ki of 980 nM. L-phenylalanine is a competitive antagonist for the glycine- and glutamate-binding sites […]

For research use only. We do not sell to patients. [Des-His1,Glu9]-Glucagon amide TFA Biological Activity：[Des-His1,Glu9]-Glucagon amide TFA is a potent and peptide antagonist of the glucagon receptor, with a pA2 of 7.2. [Des-His1,Glu9]-Glucagon amide TFA is potentially useful in the study of the pathogenesis of diabetes. Research Area：Metabolic Disease Targets：GCGR Related Screening Libraries:Bioactive Compound Library […]

For research use only. We do not sell to patients. Diphenhydramine-d6 hydrochloride CAS No. : 1189986-72-8 Biological Activity：Diphenhydramine-d6 hydrochloride is the deuterium labeled Diphenhydramine hydrochloride. Diphenhydramine hydrochloride is a first-generation histamine H1-receptor antagonist with anti-cholinergic effect. Diphenhydramine hydrochloride can across the ovine blood-brain barrier (BBB)[2]. Research Area：Inflammation/Immunology|Endocrinology Targets：Histamine Receptor|Endogenous Metabolite Related Small Molecules:D-α-Hydroxyglutaric acid disodium;Nicotinamide […]

For research use only. We do not sell to patients. Pranlukast hemihydrate CAS No. : 150821-03-7 Biological Activity：Pranlukast hemihydrate is a highly potent, selective and competitive antagonist of peptide leukotrienes. Pranlukast inhibits [3H]LTE4, [3H]LTD4, and [3H]LTC4 bindings to lung membranes with Kis of 0.63±0.11, 0.99±0.19, and 5640±680 nM, respectively. Research Area：Inflammation/Immunology Targets：Leukotriene Receptor|Endogenous Metabolite Related […]

For research use only. We do not sell to patients. SBI-115 CAS No. : 882366-16-7 Biological Activity：SBI-115 is a TGR5 (GPCR19) antagonist. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5. Research Area：Others Targets：G protein-coupled Bile Acid Receptor 1 Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Anti-Obesity Compound Library;Lipid Metabolism Compound Library […]

For research use only. We do not sell to patients. Hydroxyzine pamoate CAS No. : 10246-75-0 Biological Activity：Hydroxyzine pamoate is a histamine H1-receptor antagonist. Target: Histamine H1-Receptor Hydroxyzine inhibits carbachol (10 μM)-induced serotonin release by 34% at 10 μM, by 25% 1 μM and by 17% 0.1 μM in pretreated bladder slices for 60 min […]

For research use only. We do not sell to patients. [D-Phe2,D-Ala6]-LH-RH CAS No. : 54784-44-0 Biological Activity：[D-Phe2,D-Ala6]-LH-RH is a potent LH-RH antagonist. [D-Phe2,D-Ala6]-LH-RH shows anti-LH/FSH-RH and antiovulatory activities. Research Area：Endocrinology Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural […]

For research use only. We do not sell to patients. Rat CGRP-(8-37) CAS No. : 129121-73-9 Biological Activity：Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist. Research Area：Neurological Disease|Cardiovascular Disease Targets：CGRP Receptor Related Screening Libraries:Bioactive Compound Library Plus;Peptide Library; Related Small Molecules:Vazegepant hydrochloride;Adrenomedullin (16-31), human;MK-3207 Hydrochloride;α-CGRP, rat;Cagrilintide acetate;HTL22562;SUN B8155;Adrenomedullin (11-50), rat;Atogepant;β-CGRP, human TFA;Calcitonin (salmon);Calcitonin […]