Tag: Antagonist

For research use only. We do not sell to patients. RU 58841 CAS No. : 154992-24-2 Biological Activity：RU 58841 (PSK-3841) is a specific androgen receptor antagonist or anti-androgen. RU 58841 (PSK-3841) has a dramatic effect on hair regrowth. Research Area：Endocrinology Targets：Androgen Receptor Related Screening Libraries:Bioactive Compound Library Plus;Endocrinology Compound Library;Transcription Factor-Targeted Library;Anti-Prostate Cancer Compound Library;Nuclear […]

For research use only. We do not sell to patients. ORIC-101 CAS No. : 2222344-98-9 Biological Activity：ORIC-101 is a highly potent and selective glucocorticoid receptor antagonist, with an EC50 of 5.6 nM. Anti-cancer activity. Research Area：Cancer|Endocrinology Targets：Glucocorticoid Receptor Related Screening Libraries:Clinical Compound Library Plus;Bioactive Compound Library Plus; Related Small Molecules:Deflazacort-D5;Glucocorticoid receptor agonist-2;AZD2906;Beclometasone dipropionate;Clobetasone butyrate;Cortisone-d2;Clobetasone butyrate-d7;Cortisone-13C3;Glucocorticoid […]

For research use only. We do not sell to patients. Pipazethate CAS No. : 2167-85-3 Biological Activity：Pipazethate (SKF 70230A), a pyridobenzothiazine derivative, is a potent GABA antagonist. Pipazethate has antitussive activity. Pipazethate can be used in research in cough supressant. Research Area：Others Targets：GABA Receptor Related Small Molecules:SKF89976A hydrochloride;mGAT-IN-1;Alpidem;FG8119;Valerenic acid;Picrotoxinin;Miltirone;Etifoxine-13C,d3;Adipiplon;Gabazine;Broflanilide;Fluxametamide;ONO-8590580;γ-Aminobutyric acid-d6;Ginsenoside Rc;Fipronil;p-Hydroxybenzaldehyde-13C;Lesogaberan hydrochloride;FG 7142;Isoguvacine hydrochloride;Guvacine ethyl […]

For research use only. We do not sell to patients. PSB-0739 CAS No. : 1052087-90-7 Biological Activity：PSB-0739 is a high-affinity potent, competitive, nonselective platelet P2Y12 receptor antagonist with a Ki values of 24.9 nM. The P2Y12 receptor plays a crucial role in platelet aggregation. Antithrombotic effect. Research Area：Cardiovascular Disease Targets：P2Y Receptor Related Small Molecules:YM-254890;BPTU;Uridine 5′-diphosphoglucose […]

For research use only. We do not sell to patients. Sultopride-d5 CAS No. : 1185004-43-6 Biological Activity：Sultopride-d5 (LIN-1418-d5) is the deuterium labeled Sultopride. Sultopride (LIN-1418) is a selective antagonist of dopamine D2 receptor[2]. Research Area：Neurological Disease Targets：Dopamine Receptor Related Small Molecules:Alizapride hydrochloride;Thioproperazine;Bromopride-d3;Nuciferine;Glaucine;SB-277011 dihydrochloride;MIF-1 TFA;Sulpiride;(Rac)-Razpipadon;Clebopride malate;WAY-100635;Flupentixol-d4 dihydrochloride;Cariprazine-d6 hydrochloride;Itopride-d6 hydrochloride;ONC206;Brexpiprazole S-oxide;cis-(Z)-Flupentixol dihydrochloride;D4R antagonist-1;U91356 Trending products：Recombinant Proteins  |  […]

For research use only. We do not sell to patients. Dolasetron-d4 Biological Activity：Dolasetron-d4 is deuterium labeled Dolasetron. Research Area：Others Targets：5-HT Receptor Related Small Molecules:F 13714;Mosapride-d5;Nuciferine;Renzapride;LY 344864 racemate;Harmine hydrochloride;Valerenic acid;Arotinolol;Melitracen-d6 hydrochloride;WAY-100635;Nelotanserin;Flupentixol-d4 dihydrochloride;Cariprazine-d6 hydrochloride;Tetrahydro-β-carboline;CP-809101;Volinanserin-d4 hydrochloride;Masupirdine free base;BRL-15572 dihydrochloride;LY393558;Brexpiprazole S-oxide Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  |  PROTAC  |  Isotope-Labeled Compounds  […]

For research use only. We do not sell to patients. ALB-127158(a) CAS No. : 1173154-32-9 Biological Activity：ALB-127158(a) is a potent and selective melanin concentrating hormone 1 (MCH1) receptor antagonist. Research Area：Metabolic Disease|Endocrinology Targets：MCHR1 (GPR24) Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;Endocrinology Compound Library;Anti-Obesity Compound Library;Targeted Diversity Library; Related Small Molecules:SB-568849;[Ala17]-MCH;AZD1979;ATC0175;MCH(human, […]

For research use only. We do not sell to patients. Hydroxyzine D8 CAS No. : 1189480-47-4 Biological Activity：Hydroxyzine D8 is deuterium labeled Hydroxyzine. Hydroxyzine is a histamine H1-receptor antagonist. Research Area：Endocrinology|Inflammation/Immunology Targets：Histamine Receptor Related Screening Libraries:Bioactive Compound Library Plus; Related Small Molecules:Tripelennamine;Brompheniramine-d6 maleate;Samelisant;Chlorphenoxamine;H3 receptor-MO-1;Diphenhydramine;ABT-239;Ketotifen fumarate;Ranitidine;Cetirizine;Diphenylpyraline hydrochloride;Loratadine-d5;Phenyltoloxamine;Ritanserin;BMY-25271;FRG8701;Mecamylamine hydrochloride;Cimetidine sulfoxide;Brompheniramine maleate;Tecastemizole;Famotidine-13C,d3;Bromazine-d6 hydrochloride Trending products：Recombinant Proteins  |  Bioactive […]

For research use only. We do not sell to patients. Promethazine-d4 hydrochloride CAS No. : 1173018-74-0 Biological Activity：Promethazine-d4 hydrochloride is the deuterium labeled Promethazine hydrochloride. Promethazine hydrochloride is the first-generation antihistamine; strong antagonist of the H1 receptor and moderate mACh receptor antagonist, moderate affinity for 5-HT2A, 5-HT2C, D2 and α1-adrenergic receptors. Research Area：Neurological Disease|Endocrinology Targets：Histamine […]

For research use only. We do not sell to patients. CCR4 antagonist 3-1 CAS No. : 1957-01-3 Biological Activity：CCR4 antagonist 3 is a potent chemokine receptor 4 (CCR4) antagonist with an IC50 value of 1.7 μM for [125I]TARC (thymus and activation regulated chemokine). CCR4 antagonist 3 inhibits binding of radiolabeled TARC and macrophage-derived chemokine (MDC) […]