Tag: Antagonist

For research use only. We do not sell to patients. Oxprenoate potassium CAS No. : 76676-34-1 Biological Activity：Oxprenoate potassium is a potent mineralocorticoid (MR) antagonist. Oxprenoate potassium accentuates DEX (dexamethasone)-induced apoptosis. Research Area：Endocrinology Targets：Mineralocorticoid Receptor Related Small Molecules:Desoxycorticosterone pivalate-d8;Canrenone-d6;(S)-Baxdrostat;Canrenone-d4;18-Oxocortisol;Desoxycorticosterone pivalate;Vamorolone;Dicirenone;Osilodrostat;Balcinrenone;Lorundrostat;Esaxerenone;Deoxycorticosterone acetate;Canrenoate potassium;Ocedurenone;Apararenone;PF-3882845;Finerenone Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  […]

For research use only. We do not sell to patients. GRPR antagonist-2 Biological Activity：GRPR antagonist-2 is a potent gastrin releasing peptide receptor (GRPR) antagonist, having the cytotoxicity against certain cancer cells (IC50 of 0.77 and 2.5 μM in HGC-27 and Pan02 cells, respectively). Anticancer activity. Research Area：Cancer Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin […]

For research use only. We do not sell to patients. A1AR antagonist 3 CAS No. : 2413257-73-3 Biological Activity：A1AR antagonist 3 (compound 13) is a selective adenosine 1 (A1) receptor antagonist with Kis of 9.69 nM and 0.529 nM for human A1 and rat A1, respectively. A1AR antagonist 3 can be used for researching neurological […]

For research use only. We do not sell to patients. MRS1186 CAS No. : 183721-03-1 Biological Activity：MRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM. Research Area：Inflammation/Immunology Targets：Adenosine Receptor Related Small Molecules:MRS 1523;APNEA;MIPS521;Derenofylline;FSCPX;Theobromine-d3;Inosine-13C;Norisoboldine;N-0861 racemate;Xanthine amine congener dihydrochloride;LUF6096;A1/A3 AR antagonist 1;ATL-801;Istradefylline;Doxofylline-d6;A1AR antagonist 3;A2A/A3 AR antagonist-1;A2AAR/HDAC-IN-2;MRS-1191;MRS5698;GP531;Imaradenant;PSB-0788 Trending products：Recombinant Proteins  […]

For research use only. We do not sell to patients. Chlorpheniramine-d4 maleate CAS No. : 2747915-71-3 Biological Activity：Chlorpheniramine-d4 (maleate) is deuterium labeled Chlorpheniramine (maleate). Research Area：Inflammation/Immunology|Endocrinology Targets：Histamine Receptor Related Small Molecules:Tripelennamine;Brompheniramine-d6 maleate;Samelisant;Chlorphenoxamine;H3 receptor-MO-1;Diphenhydramine;ABT-239;Ketotifen fumarate;Ranitidine;Cetirizine;Diphenylpyraline hydrochloride;Loratadine-d5;Phenyltoloxamine;Ritanserin;BMY-25271;FRG8701;Mecamylamine hydrochloride;Cimetidine sulfoxide;Brompheniramine maleate;Tecastemizole;Famotidine-13C,d3;Bromazine-d6 hydrochloride Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  Fluorescent Dye  |  PROTAC  |  […]

For research use only. We do not sell to patients. PHTPP CAS No. : 805239-56-9 Biological Activity：PHTPP is a selective estrogen receptor β (ERβ) antagonist with 36-fold selectivity over ERα. Research Area：Cancer Targets：Estrogen Receptor/ERR Related Screening Libraries:Bioactive Compound Library Plus;Anti-Cancer Compound Library;Anti-Breast Cancer Compound Library;Human Metabolite Library;Nuclear Receptor Compound Library; Related Small Molecules:DS20362725;LSD1/ER-IN-1;Giredestrant;Avobenzone;Estriol-d3;Chrysin;ERRγ Inverse Agonist […]

For research use only. We do not sell to patients. L-Phenylalanine-13C6 CAS No. : 180268-82-0 Biological Activity：L-Phenylalanine-13C6 ((S)-2-Amino-3-phenylpropionic acid-13C6) is the 13C-labeled L-Phenylalanine. L-Phenylalanine ((S)-2-Amino-3-phenylpropionic acid) is an essential amino acid isolated from Escherichia coli. L-Phenylalanine is a α2δ subunit of voltage-dependent Ca+ channels antagonist with a Ki of 980 nM. L-phenylalanine is a competitive […]

For research use only. We do not sell to patients. CYN 154806 CAS No. : 183658-72-2 Biological Activity：CYN 154806, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively[2]. Research Area：Endocrinology Targets：Somatostatin […]

For research use only. We do not sell to patients. SCH 546738 CAS No. : 906805-42-3 Biological Activity：SCH 546738 is a potent, orally active and non-competitive CXCR3 antagonist, the affinity constant (Ki) of SCH 546738 binding to human CXCR3 receptor is determined to be 0.4 nM in multiple experiments. Research Area：Inflammation/Immunology|Endocrinology Targets：CXCR Related Screening Libraries:Bioactive […]

For research use only. We do not sell to patients. Alprenolol-d7 hydrochloride CAS No. : 2714410-80-5 Biological Activity：Alprenolol-d7 ((RS)-Alprenolol-d7) hydrochloride is the deuterium labeled Alprenolol hydrochloride. Alprenolol hydrochloride is a non-selective beta blocker as well as 5-HT1A receptor antagonist. Research Area：Cancer Targets：5-HT Receptor Related Small Molecules:F 13714;Mosapride-d5;Nuciferine;Renzapride;LY 344864 racemate;Harmine hydrochloride;Valerenic acid;Arotinolol;Melitracen-d6 hydrochloride;WAY-100635;Nelotanserin;Flupentixol-d4 dihydrochloride;Cariprazine-d6 hydrochloride;Tetrahydro-β-carboline;CP-809101;Volinanserin-d4 hydrochloride;Masupirdine […]