Palonidipine

For research use only. We do not sell to patients. Palonidipine CAS No. : 96515-73-0 Biological Activity:Palonidipine is a calcium antagonist which is potential for the therapy of angina-pectoris and hypertension[2][3]. Research Area:Cardiovascular Disease Targets:Calcium Channel Related Small Molecules:Benidipine hydrochloride;CaV1.3 antagonist-1;14-Deoxyandrographolide;(Rac)-MEM 1003;Glaucine;Efonidipine hydrochloride monoethanolate;L-Ascorbic acid sodium salt;Brompheniramine-d6 maleate;MRS 1523;Nilvadipine;Lercanidipine;CP-060;Anipamil-d25 hydrochloride;ISX-9;ω-Conotoxin MVIIC;Catharanthine;Thapsigargin;Tetrandrine;Ginsenoside Rd;Manidipine dihydrochloride;ω-Agatoxin IVA;AE0047 Hydrochloride;PDE1-IN-4 […]

SB 204741

For research use only. We do not sell to patients. SB 204741 CAS No. : 152239-46-8 Biological Activity:SB 204741 is a selective and high affinity 5-HT2B antagonist with a pKi value of 7.1. Research Area:Cardiovascular Disease Targets:5-HT Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;Anti-Cardiovascular Disease Compound Library;Ferroptosis Compound Library;Neurotransmitter […]

Vapreotide acetate

For research use only. We do not sell to patients. Vapreotide acetate CAS No. : 849479-74-9 Biological Activity:Vapreotide acetate (RC-160 acetate; BMY-41606 acetate) is a neurokinin-1 (NK1) receptor antagonist, with an IC50 of 330 nM. Research Area:Cancer Targets:Neurokinin Receptor Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;GPCR/G […]

SB-200646

For research use only. We do not sell to patients. SB-200646 CAS No. : 143797-63-1 Biological Activity:SB-200646 is the first selective 5-HT2B/2C over 5-HT2A receptor antagonist with pKi values of 7.5, 6.9 and 5.2 for 5-HT2B, 5-HT2C and 5-HT2A, respectively. SB-200646 is orally active and has electrophysiological and anxiolytic properties in vivo[2]. Research Area:Neurological Disease […]

Rislenemdaz

For research use only. We do not sell to patients. Rislenemdaz CAS No. : 808732-98-1 Biological Activity:Rislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC 50 of 8.1 nM and 3.6 nM, respectively. Research Area:Neurological Disease Targets:iGluR Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound […]

CAY10471 Racemate

For research use only. We do not sell to patients. CAY10471 Racemate CAS No. : 844639-57-2 Biological Activity:CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist, with a Ki of 0.6 nM for hCRTH2, selective over human thromboxane A2 receptor TP (Ki, >10000 nM) or PGD2 receptor DP (Ki, […]

BE1218

For research use only. We do not sell to patients. BE1218 Biological Activity:BE1218 is a liver X receptor (LXR) inverse agonist with IC50 values of 9 nM and 7 nM against LXRα and LXRβ, respectively. Research Area:Cancer Targets:LXR Related Small Molecules:XL041;DMHCA;Saikosaponin A;27-Hydroxycholesterol;LXRβ agonist-3;RGX-104;24(S)-Hydroxycholesterol;SR9238;BMS-779788;SR9243;AZ876;T0901317;LXRβ agonist-2;GSK2033;LXR antagonist 2;LXR agonist 1;GW3965;LXR-623;Nagilactone B;LXR agonist 2;Rovazolac;GSK3987 Trending products:Recombinant Proteins  |  […]

ABP688

For research use only. We do not sell to patients. ABP688 CAS No. : 924298-51-1 Biological Activity:ABP688 is a high affinity human mGluR5 antagonist with anKi of 1.7 nM. Radioisotope-labeled ABP688 can be used as a PET tracer for clinical imaging of the mGlu5 receptor. Research Area:Others Targets:mGluR Related Small Molecules:LY3020371 hydrochloride;ZJ43;FPTQ;(S)-MCPG;mGluR2 modulator 1;VU6010572;Mavoglurant racemate;DFMTI;JNJ16259685;Auglurant;FITM;(-)-Camphoric […]

Yamogenin

For research use only. We do not sell to patients. Yamogenin CAS No. : 512-06-1 Biological Activity:Yamogenin (Neodiosgenin) is a diastereomer of diosgenin. Yamogenin (Neodiosgenin) antagonizes the activation of the liver X receptor (LXR) in luciferase ligand assay. Yamogenin (Neodiosgenin) inhibits triacylglyceride (TG) accumulation through the suppression of gene expression of fatty acid synthesis in […]

IPSU

For research use only. We do not sell to patients. IPSU CAS No. : 1373765-19-5 Biological Activity:IPSU is a selective, orally available and brain penetrant OX2R antagonist with a pKi of 7.85. Research Area:Neurological Disease|Endocrinology Targets:Orexin Receptor (OX Receptor) Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;Endocrinology Compound Library;Orally Active Compound […]