Tag: Activator

For research use only. We do not sell to patients. 5(S)15(S)-DiHETE CAS No. : 82200-87-1 Biological Activity：5(S)15(S)-DiHETE is an “activated” intermediate, inhibits platelet aggregation with an IC50 of 1.3 μM. 5(S)15(S)-DiHETE enhances the rate of either LXA4 or LXB4 biosynthesis. Research Area：Inflammation/Immunology|Cardiovascular Disease Targets：Interleukin Related Related Small Molecules:AX-024;Ginsenoside F3;Perakizumab;PNRI-299;CTX-471;Ac-YVAD-CHO;Deucravacitinib;Mulberroside A;NFAT Transcription Factor Regulator-1;IL-17A antagonist 1;Kansuinine […]

For research use only. We do not sell to patients. LM22B-10 CAS No. : 342777-54-2 Biological Activity：LM22B-10 is an activator of TrkB/TrkC neurotrophin receptor, and can induce TrkB, TrkC, AKT and ERK activation in vitro and in vivo. Research Area：Neurological Disease Targets：Akt|Trk Receptor|ERK Related Screening Libraries:Bioactive Compound Library Plus;Immunology/Inflammation Compound Library;Kinase Inhibitor Library;MAPK Compound Library;Neuronal […]

For research use only. We do not sell to patients. Grape seed extract CAS No. : 84929-27-1 Biological Activity：Grape seed extract is a natural product, with anti-inflammatory and anti-proliferative effects. Grape seed extract shows inhibitory activity on the fat-metabolizing enzymes pancreatic lipase and lipoprotein lipase. Grape seed extract induces apoptotic in human colorectal cancer cells[2][3]. […]

For research use only. We do not sell to patients. cGAMP CAS No. : 849214-04-6 Biological Activity：cGAMP (Cyclic GMP-AMPP) functions as an endogenous second messenger in metazoans and triggers interferon production in response to cytosolic DNA. cGAMP activates stimulator of interferon genes (STING), which activates a signaling cascade leading to the production of type I […]

For research use only. We do not sell to patients. GLUT4 activator 1 CAS No. : 2253733-37-6 Biological Activity：GLUT4 activator 1 (Compound 26b) is a potent glucose transporter type 4 (GLUT4) translocation activator with an EC50 of 0.14 μM. Research Area：Metabolic Disease Targets：GLUT Related Screening Libraries:Bioactive Compound Library Plus; Related Small Molecules:Sennidin A;Licarin B;GLUT4-IN-2;STF-31;KPH2f;BAY-876;MOTS-c(human) acetate;Phloretin;GLUT […]

For research use only. We do not sell to patients. CLEFMA CAS No. : 1246964-32-8 Biological Activity：CLEFMA is a curcuminoid with antitumor activity. CLEFMA inhibits tumor growth is associated with NF-κB-regulated anti-inflammatory and anti-metastatic effects[2]. Research Area：Cancer Targets：Apoptosis Related Small Molecules:Physalin A;Bomedemstat ditosylate;Enpp/Carbonic anhydrase-IN-1;GK563;Calpeptin;Lobetyolin;BJE6-106;Dinaciclib;Ecteinascidin 770;MDM2-p53-IN-15;AT9283;Staurosporine;SNS-032;C188-9;ZLDI-8;Topoisomerase I/II inhibitor 3;Xevinapant;Mangiferin;Cambinol;Antioxidant agent-5;Apoptosis inducer 9;Bafetinib;Cyclovirobuxine D;STAT3-IN-10;Rigosertib sodium Trending products：Recombinant […]

For research use only. We do not sell to patients. Melengestrol acetate-d2 Biological Activity：Melengestrol acetate-d2 is the deuterium labeled Melengestrol acetate. Melengestrol acetate is a progesterone derivative, acts as an orally active corticosteroid hormone to promote endometrial proliferation, pregnancy maintenance, and delay of menstrual activity. Melengestrol Acetate is used as a contraceptive agent for growth […]

For research use only. We do not sell to patients. Coluracetam CAS No. : 135463-81-9 Biological Activity：Coluracetam(MKC-231) is a new choline uptake enhancer. IC50 value: Target: in vitro: MKC-231 (10(-10)-10(-6) moll) significantly increased high affinity choline uptake (HACU) when it was incubated with the hippocampal synaptosomes of ethylcholine mustard aziridinium ion (AF64A) treated rats, but […]

For research use only. We do not sell to patients. (24R)-MC 976 CAS No. : 112828-09-8 Biological Activity：(24R)-MC 976 is a Vitamin D3 derivative. Research Area：Metabolic Disease Targets：VD/VDR Related Small Molecules:Atocalcitol;VD3-d6;Dihydrotachysterol;Tacalcitol;Impurity F of Calcipotriol;MeTC7;VDR agonist 1;TEI-9648;CB1151;MC 1046;1alpha, 25-Dihydroxy VD2-13C2;Secalciferol;5,6-trans-Vitamin D3;Chol-5-en-24-al-3β-ol;Maxacalcitol-d6;Vitamin D3-13C3;Vitamin D3-D7;Vitamin D4;Vitamin D2-d6 Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  Natural Products  |  […]

For research use only. We do not sell to patients. β-Pompilidotoxin TFA Biological Activity：β-Pompilidotoxin TFA (β-PMTX TFA), a wasp venom, can slow sodium channel inactivation and increases steady-state sodium current in cells. Research Area：Neurological Disease Targets：Sodium Channel Related Small Molecules:Lu AE98134;Zandatrigine;Veratridine;Brompheniramine-d6 maleate;GX-674;Dibucaine;Sodium Channel inhibitor 2;3-Deoxyaconitine;20(S)-Ginsenoside Rg3;Tocainide hydrochloride;Licarbazepine-d4-1;Metaflumizone-d4;β-Pompilidotoxin;Nav1.1 activator 1;ICA-121431;Brompheniramine maleate;ABBV-318;PF 05089771;DPI 201-106;TC-N 1752 Trending products：Recombinant […]