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Rosiglitazone maleate
CAS No. : 155141-29-0
Biological Activity：Rosiglitazone maleate (BRL 49653C) is a potent and selective activator of PPARγ, with EC50s of 30 nM, 100 nM and 60 nM for PPARγ1, PPARγ2, and PPARγ, respectively, and a Kd of appr 40 nM for PPARγ; Rosiglitazone maleate is also an modulator of TRP channels, inhibits TRP melastatin 2 (TRPM2), TRPM3 and activates TRP canonical 5 (TRPC5).
Research Area：Cancer|Metabolic Disease|Inflammation/Immunology
Targets：Ferroptosis|Autophagy|TRP Channel|PPAR
Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library Plus;Apoptosis Compound Library;Cell Cycle/DNA Damage Compound Library;Immunology/Inflammation Compound Library;Membrane Transporter/Ion Channel Compound Library;Neuronal Signaling Compound Library;FDA-Approved Drug Library;Anti-Cancer Compound Library;Antiviral Compound Library;Autophagy Compound Library;Anti-Aging Compound Library;Drug Repurposing Compound Library;Anti-diabetic Compound Library;Oxygen Sensing Compound Library;Ferroptosis Compound Library;Anti-COVID-19 Compound Library;NMPA-Approved Drug Library;FDA Approved & Pharmacopeial Drug Library;Drug-Induced Liver Injury (DILI) Compound Library;Anti-Obesity Compound Library;Transcription Factor-Targeted Library;Lipid Metabolism Compound Library ;Mechanoreceptors Compound Library;Targeted Diversity Library;Rare Diseases Drug Library;Antidepressant Compound Library;EMA-Approved Drug Library;FDA-Approved Anticancer Drug Library;Human Metabolite Library;Anti-Prostate Cancer Compound Library;Nuclear Receptor Compound Library;Non-steroidal Anti-Inflammatory Compound Library;Osteogenesis Compound Library;Cancer Stem Cells Compound Library;
Related Small Molecules:V116517;CIL56;DB0614;GSK2332255B;Pregnenolone monosulfate sodium;Ciclopirox-d11;Ciclopirox olamine;Curcumin;TRPC5-IN-4;OptoBI-1;Falcarindiol;5-Aminosalicylic Acid-D3 hydrochloride;Retinoic acid;SB-705498;PPARγ agonist 7;TRPC3/6-IN-1;ABT-239;Pyr3;Licarin B;Asivatrep;(-)-Epicatechin;Mifobate;Eugenol-d3
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