Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. Uralenol CAS No. : 139163-15-8 Biological Activity：Uralenol is a natural PTP1B inhibitor (IC50=21. 5 μM) from Broussonetia papyrifera. PTP1B have been shown to play a major role in the dephosphorylation of the insulin receptor in many cellular and biochemical studies. Research Area：Metabolic Disease Targets：Phosphatase Related […]
For research use only. We do not sell to patients. Levobetaxolol CAS No. : 93221-48-8 Biological Activity：Levobetaxolol is a potent and high affinity β-adrenergic antagonist with IC50 values of 33.2, 2970, 709 nM for guinea pig atrial β1, tracheal β2 and rat colonic β3 receptors, respectively. Levobetaxolol reduces IOP (intraocular pressure). Levobetaxolol exhibits a micromolar […]
For research use only. We do not sell to patients. SulfoxFluor CAS No. : 2143892-50-4 Biological Activity：SulfoxFluor is a novel deoxyfluorination reagent. SulfoxFluor is shelf-stable, easy-to-handle, fluorine-economical, and highly selective. Research Area：Others Targets：Others Related Screening Libraries:Bioactive Compound Library Plus; Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending […]
For research use only. We do not sell to patients. GATA4-NKX2-5-IN-1 CAS No. : 544681-96-1 Biological Activity：GATA4-NKX2-5-IN-1 (Compound 3) dose-dependently inhibits the GATA4–NKX2-5 transcriptional synergy with an IC50 of 3 μM. GATA4-NKX2-5-IN-1 exhibits no activity on the protein kinases involved in the regulation of GATA4 phosphorylation, and it modulates the hypertrophic agonist-induced cardiac gene expression. […]
For research use only. We do not sell to patients. Amoxapine CAS No. : 14028-44-5 Biological Activity：Amoxapine is a tetracyclic antidepressant of the dibenzoxazepine family, though it is often classified as a secondary amine tricyclic antidepressant. Research Area：Neurological Disease Targets：Others Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug Library Plus;FDA-Approved Drug Library Mini;Bioactive Compound Library […]
For research use only. We do not sell to patients. BIX-01294 CAS No. : 935693-62-2 Biological Activity：BIX-01294 is a reversible and highly selective G9a and GLP Histone Methyltransferase inhibitor, with IC50s of of 1.7 μM and 0.9 μM, respectively. BIX-01294 inhibits G9a/GLP by competing for binding with the amino acids N-terminal of the substrate lysine […]
For research use only. We do not sell to patients. 2-Amino-3-mercaptopropanoic acid hydrochloride hydrate CAS No. : 96998-61-7 Biological Activity：2-Amino-3-mercaptopropanoic acid hydrochloride hydrate is a cysteine derivative. Research Area：Others Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products […]
For research use only. We do not sell to patients. DBCO-PEG6-amine TFA Biological Activity：DBCO-PEG6-amine TFA is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs. Research Area：Others Targets：PROTAC Linkers Related Small Molecules:N-(Mal-PEG6)-N-bis(PEG7-TCO);Propargyl-PEG2-CH2COOH;NHS ester-PEG10-COOH;Tos-PEG5-Boc;Bis-PEG6-NHS ester;Azide-PEG12-alcohol;Fmoc-PEG6-NHS ester;Boc-C1-PEG3-C4-OBn;Boc-NH-PEG8-C2-Br;Propargyl-PEG14-Boc;m-PEG21-OH;Bromo-PEG3-THP;m-PEG8-Ms;Bis-PEG10-NHS ester;TCO-PEG3-acid;m-PEG8-DBCO;Azide-PEG6-Tos;Acid-PEG3-C2-Boc;m-PEG-mal (MW 2000);Benzyl-PEG7-t-butyl ester;Boc-Pip-alkyne-Ph-COOH;Biotin-PEG2-C6-azide;Bis-PEG4-acid;Active-mono-sulfone-PEG8-acid;Br-PEG6-C2-NHBoc;HO-PEG8-CH2COOH;NH2-PEG4-CH2CH2COOH;N-(Propargyl-PEG2)-N-Boc-PEG3-t-butyl ester;Bromoacetamido-PEG8-Boc;Carboxy-PEG2-sulfonic acid Trending products：Recombinant Proteins | Bioactive Screening Libraries | Natural Products […]
For research use only. We do not sell to patients. β-Amyloid (1-42), (rat/mouse) (TFA) Biological Activity：β-Amyloid (1-42), (rat/mouse) TFA is a 42-aa peptide, shows cytotoxic effect on acute hippocampal slices, and used in the research of Alzheimer’s disease. Research Area：Neurological Disease Targets：Amyloid-β Related Screening Libraries:Bioactive Compound Library Plus;Peptide Library; Related Small Molecules:β-Amyloid (13-27);Saikosaponin C;β-Amyloid (12-28) […]
For research use only. We do not sell to patients. L-Thyroxine sodium CAS No. : 55-03-8 Biological Activity：L-Thyroxine sodium (Levothyroxine sodium) is a synthetic hormone for the research of hypothyroidism. DIO enzymes convert biologically active thyroid hormone (Triiodothyronine,T3) from L-Thyroxine (T4). Research Area：Endocrinology|Cancer Targets：Thyroid Hormone Receptor|Endogenous Metabolite Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug […]