Master of Bioactive Molecules | Inhibitors, Screening Libraries & Proteins
For research use only. We do not sell to patients. Dinaciclib CAS No. : 779353-01-4 Biological Activity：Dinaciclib (SCH 727965) is a potent inhibitor of CDK, with IC50s of 1 nM, 1 nM, 3 nM, and 4 nM for CDK2, CDK5, CDK1, and CDK9, respectively. Research Area：Cancer Targets：CDK|Apoptosis Related Screening Libraries:Drug Repurposing Compound Library Plus;FDA-Approved Drug […]
For research use only. We do not sell to patients. VEGFR-2-IN-24 CAS No. : 2455414-26-1 Biological Activity：VEGFR-2-IN-24 is a potent VEGFR-2 inhibitor with IC50 value of 0.22 µM. VEGFR-2-IN-24 can be used for tumor research. Research Area：Cancer Targets：VEGFR Related Small Molecules:(Z)-FeCP-oxindole;BMS-690514;PROTAC VEGFR-2 degrader-2;Henatinib;PI3K/VEGFR2-IN-1;Hydroxytanshinone IIA;Chiauranib;Foretinib;ZM323881 hydrochloride;PTC299;ENMD-2076 Tartrate;Aflibercept;SU5408;MAZ51;R1530;AZD2932;R916562;XL092;Tyrosine kinase-IN-1;DMH4;Bucillamine Trending products：Recombinant Proteins | Bioactive Screening Libraries | […]
For research use only. We do not sell to patients. WKYMVM CAS No. : 187986-17-0 Biological Activity：WKYMVM is a potent N-formyl peptide receptor (FPR1) and FPRL1/2 agonist, also activates several leukocyte effector functions such as chemotaxis, mobilization of complement receptor-3, and activation of the NADPH oxidase[2]. Research Area：Inflammation/Immunology Targets：Formyl Peptide Receptor (FPR) Related Screening Libraries:Bioactive […]
For research use only. We do not sell to patients. Anhydrosafflor yellow B CAS No. : 184840-84-4 Biological Activity：Anhydrosafflor yellow B (AHSYB) is a quinochalcone C-glycoside isolated from Carthamus tinctorius. Anhydrosafflor yellow B inhibits ADP-induced platelet aggregation, exhibits significant anti-oxidative effects in vitro, and possesses certain activity against H2O2-induced cytotoxicity in cultured PC12 cells and […]
For research use only. We do not sell to patients. RP-64477 CAS No. : 135239-65-5 Biological Activity：RP-64477 is a potent inhibitor of the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT). Research Area：Cardiovascular Disease Targets：Acyltransferase Related Screening Libraries:Bioactive Compound Library Plus;Metabolism/Protease Compound Library;Anti-Cardiovascular Disease Compound Library;Lipid Metabolism Compound Library ; Related Small Molecules:Enniatin A;IWP-12;ABT-046;PF-04620110;ACAT-IN-5;TP-020;Diacylglycerol acyltransferase inhibitor-1;JNJ-DGAT2-A;DGAT-1 […]
For research use only. We do not sell to patients. Regorafenib-13C,d3 Biological Activity：Regorafenib-13C,d3 is the 13C- and deuterium labeled Regorafenib. Regorafenib (BAY 73-4506) is a multi-targeted receptor tyrosine kinase inhibitor with IC50s of 13/4.2/46, 22, 7, 1.5 and 2.5 nM for VEGFR1/2/3, PDGFRβ, Kit, RET and Raf-1, respectively. Research Area：Cancer Targets：Autophagy|Raf|VEGFR|RET|PDGFR Related Small Molecules:(Z)-FeCP-oxindole;Avutometinib;VEGFR-2-IN-24;BMS-690514;PROTAC VEGFR-2 […]
For research use only. We do not sell to patients. Haloprogin CAS No. : 777-11-7 Biological Activity：Haloprogin is a potent antifungal agent. Haloprogin has activity against dermatophytes, Candida spp and a limited number of Gram-positive bacteria. Research Area：Infection Targets：Fungal Related Small Molecules:Antifungal agent 20;Debneyol;Staurosporine;Ciclopirox-d11;Ciclopirox olamine;Clotrimazole-d5;(R)-Camptothecin-d5;Ticlatone;Aminothiazole;Magnesium silicate;α-Terpinene;Hydroxyphenyllactic acid;Iprobenfos;Chlorphenesin;Moniliformin sodium salt;HLF1-11;β-Amyrin acetate;Bifonazole;Aszonapyrone A;Oenothein B;Pyrimorph;(+)-Magnoflorine iodide;Antifungal agent 39 […]
For research use only. We do not sell to patients. Polyketide synthase 13-IN-1 CAS No. : 2345638-96-0 Biological Activity：Polyketide synthase 13-IN-1 (compound 32) is a polyketide synthase 13 inhibitor. Research Area：Infection|Inflammation/Immunology Targets：Others Related Small Molecules:Immune initiator-1;Obiltoxaximab;DIBAC-GGFG-NH2CH2-Dxd;Cyanine5.5 maleimide chloride;Cymarin;Z-Glycine;2-Deoxy-2-fluoro-D-glucose-13C,d7;Water-18O;Fmoc-N-Me-D-Ala-OH;3,5-Diiodo-L-tyrosine;N3-Pen-Dde;Zimeldine-d6;Ornidazole diol;Nylidrin hydrochloride;PFI-653;N-Arachidonoyl Taurine-d4;OVA Peptide (323-339);((3-Fluorophenyl)sulfonyl)glycine;7ß-Hydroxycholesterol-d7;MALAT1-IN-1;Sibiricose A1;Mefruside-d3;Ethacrynic acid mercapturate-d3;FLAG peptide;Neocurdione Trending products：Recombinant Proteins | Bioactive Screening Libraries | […]
For research use only. We do not sell to patients. trans-Cevimeline hydrochloride CAS No. : 107220-29-1 Biological Activity：Trans-Cevimeline (AF102A) (hydrochloride), as a trans-isomer of AF102B, is a M1 selective cholinergic agonist. Trans-Cevimeline (AF102A) (hydrochloride) can be used for the research of Alzheimer’s disease. Research Area：Neurological Disease Targets：mAChR Related Small Molecules:VU0357017 hydrochloride;TBPB;Imidafenacin;Sabcomeline;MK-6884;Brompheniramine-d6 maleate;Navafenterol saccharinate;DREADD agonist 21;Cyclobuxine […]
For research use only. We do not sell to patients. PXS-4728A CAS No. : 1478364-68-9 Biological Activity：PXS-4728A (BI-1467335) is a selective, orally active inhibitor of semicarbazide-sensitive amine oxidase (SSAO). PXS-4728A ameliorates chronic obstructive pulmonary disease in mice. Research Area：Inflammation/Immunology Targets：Monoamine Oxidase Related Screening Libraries:Drug Repurposing Compound Library Plus;Clinical Compound Library Plus;Bioactive Compound Library Plus;Immunology/Inflammation Compound […]