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CAS No. : 1221186-53-3

Biological Activity:TEPP-46 (ML-265) is a potent and selective pyruvate kinase M2 (PKM2) activator with an AC50 of 92 nM, showing little or no effect on PKM1, PKL and PKR.

Research Area:Cancer

Targets:Pyruvate Kinase

Related Screening Libraries:Bioactive Compound Library Plus;Kinase Inhibitor Library;Metabolism/Protease Compound Library;Anti-Cancer Compound Library;Glycolysis Compound Library;Pyroptosis Compound Library;Anti-Cancer Metabolism Compound Library;Glucose Metabolism Compound Library;Targeted Diversity Library;

Related Small Molecules:Etavopivat;Alkannin;PKM2-IN-3;PKM2-IN-1;PKM2 activator 3;PKR-IN-2;PKR activator 2;PKM2 activator 5;Mitapivat;FX-11;PKM2 activator 4;DASA-58;TEPC466;PKM2 activator 2;PKR activator 1

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