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CAS No. : 1137868-52-0

Biological Activity:TAK-960 is an orally available, selective inhibitor of polo-like kinase 1 (PLK1), with an IC50 of 0.8 nM. TAK-960 also shows inhibitory activities against PLK2 and PLK3, with IC50s of 16.9 and 50.2 nM, respectively. TAK-960 inhibits proliferation of multiple cancer cell lines and exhibits significant efficacy against multiple tumor xenografts.

Research Area:Cancer

Targets:Polo-like Kinase (PLK)

Related Screening Libraries:Clinical Compound Library Plus;Bioactive Compound Library Plus;Cell Cycle/DNA Damage Compound Library;Kinase Inhibitor Library;Anti-Cancer Compound Library;Clinical Compound Library;Anti-Aging Compound Library;Orally Active Compound Library;

Related Small Molecules:Rigosertib sodium;Centrinone;HMN-176;(1E)-CFI-400437 dihydrochloride;Poloxin;PLK1-IN-2;PLK1-IN-4;MLN0905;TC-S 7005;PLK4-IN-3;SBE13 Hydrochloride;CFI-400437;Plogosertib;Volasertib;3MB-PP1;Wortmannin;PLK1/BRD4-IN-1;Poloxime;Poloppin;Cyclapolin 9;ON1231320;BI 2536

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