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PCI 29732
CAS No. : 330786-25-9
Biological Activity：PCI 29732 is a potent, orally active, reversible BTK inhibitor with Kiapp values of 8.2, 4.6, and 2.5 nM for BTK, Lck and Lyn, respectively. PCI 29732 shows only modest inhibitory activity against Itk, another Tec family kinase. PCI 29732 inhibits the function of ABCG2 by competitively binding to the ATP-binding site of ABCG2[2].
Research Area：Inflammation/Immunology
Targets：Btk|BCRP
Related Screening Libraries:Covalent Screening Library Plus;Bioactive Compound Library Plus;Immunology/Inflammation Compound Library;Kinase Inhibitor Library;Membrane Transporter/Ion Channel Compound Library;Protein Tyrosine Kinase Compound Library;Covalent Screening Library;Orally Active Compound Library;Anti-Blood Cancer Compound Library;Cancer Stem Cells Compound Library;
Related Small Molecules:JAK3/BTK-IN-1;Elsubrutinib;ARQ 531;PF-06250112;Triclabendazole sulfoxide;Elacridar;CHMFL-EGFR-202;Avitinib;RN486;P-gp/BCRP-IN-1;GDC-0834 Racemate;Spebrutinib besylate;Vecabrutinib;BMX-IN-1;Tolebrutinib;YHO-13351;BTK-IN-16;CP-100356 hydrochloride;PD166326;(R)-Zanubrutinib;Pirtobrutinib;CTA056;Fumitremorgin C;UR-MB108;EGFR-IN-40
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