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BMS-193885
CAS No. : 186185-03-5
Biological Activity：BMS-193885 is a potent, selective, competitive, and brain penetrant neuropeptide Y1 receptor antagonist with a Ki of 3.3 nM, and has an IC50 of 5.9 nM for hY1, which displays > 100, > 160, > 160 and > 160-fold selectivity over α1, hY2, hY4 and hY5 receptors, respectively [2].
Research Area：Neurological Disease|Endocrinology
Targets：Neuropeptide Y Receptor
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Related Small Molecules:[D-Trp34]-Neuropeptide Y TFA;Pancreatic Polypeptide, human;Peptide YY (PYY), human;JNJ-5207787;[Leu31,Pro34]-Neuropeptide Y(human,rat) TFA;GR231118 TFA;Neuropeptide Y (human);RF9 hydrochloride;M1145;Galanin Receptor Ligand M35 TFA;Neuropeptide Y (3-36) (porcine);CART (55-76), rat;Galantide;RFRP-3(human) TFA;BIBO3304 TFA;Neuropeptide SF(mouse,rat);Galanin (1-16), mouse, porcine, rat;FR252384;Galnon;[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide;CART (1-39), Human, Rat;Neuropeptide Y (13-36), amide, human;Neuropeptide S(Rat);Neuropeptide Y (22-36);Lu AA33810;Neuropeptide Y (3-36) (human, rat)
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