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MSC-4381
CAS No. : 2445185-57-7
Biological Activity：MSC-4381 (MCT4-IN-1) is an orally active and selective monocarboxylate transporter 4 (MCT4/SLC16A3) inhibitor with an IC50 of 77 nM and a Ki of 11 nM. MSC-4381 targets to the cytosolic domain of MCT4. MSC-4381 results in lactate efflux inhibition and reduction of cellular viability in MCT4 high expressing cells. MSC-4381 has the potential for MCT4 transporter inhibition research.
Research Area：Cancer
Targets：Monocarboxylate Transporter
Related Screening Libraries:Bioactive Compound Library Plus;Membrane Transporter/Ion Channel Compound Library;Anti-Cancer Compound Library;Orally Active Compound Library;Anti-Cancer Metabolism Compound Library;
Related Small Molecules:α-Cyano-4-hydroxycinnamic acid;AR-C141990 hydrochloride;MCT1-IN-2;Silychristin;AR-C155858;7ACC2;AZD3965;BAY-8002;7ACC1;Syrosingopine;VB124
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