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L-371,257
CAS No. : 162042-44-6
Biological Activity：L-371,257 is an orally bioavailable, non-blood-brain barrier penetrant, selective and competitive antagonist of oxytocin receptor (pA2=8.4) with high affinity at both the oxytocin receptor (Ki=19 nM) and vasopressin V1a receptor (Ki=3.7 nM)[2].
Research Area：Endocrinology
Targets：Oxytocin Receptor|Vasopressin Receptor
Related Screening Libraries:Bioactive Compound Library Plus;
Related Small Molecules:Lixivaptan;Mozavaptan hydrochloride;Balovaptan;Big Endothelin-1 (1-38), human;WAY-151932;Felypressin;Antagonist G TFA;Mozavaptan-d6;SKF 100398;L-368,899 hydrochloride;L-372662;Fedovapagon;Epelsiban;OT antagonist 1;Argipressin;D[LEU4,LYS8]-VP;d[Cha4]-AVP;RG7713;TASP0390325;OT-R antagonist 2;Terlipressin-d5
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