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CAS No. : 251303-04-5

Biological Activity:Ertiprotafib is an inhibitor of PTP1B, IkB kinase β (IKK-β), and a dual PPARα and PPARβ agonist, with an IC50 of 1.6 μM for PTP1B, 400 nM for IKK-β, an EC50 of ~1 μM for PPARα/PPARβ.

Research Area:Metabolic Disease


Related Screening Libraries:Bioactive Compound Library Plus;Cell Cycle/DNA Damage Compound Library;Immunology/Inflammation Compound Library;Kinase Inhibitor Library;Metabolism/Protease Compound Library;NF-κB Signaling Compound Library;Stem Cell Signaling Compound Library;Anti-Aging Compound Library;Differentiation Inducing Compound Library;Anti-diabetic Compound Library;Phosphatase Inhibitor Library;Anti-Obesity Compound Library;Transcription Factor-Targeted Library;Lipid Metabolism Compound Library ;Anti-Liver Cancer Compound Library ;Antidepressant Compound Library;Anti-Prostate Cancer Compound Library;Nuclear Receptor Compound Library;

Related Small Molecules:GNF362;ZLDI-8;Uralenol;Falcarindiol;5-Aminosalicylic Acid-D3 hydrochloride;Retinoic acid;PS-1145;SHP504;PPARγ agonist 7;Trimyristin;SHP099 hydrochloride;NF-κB-IN-1;MY10;Licarin B;Mifobate;PTP1B-IN-3 diammonium;Resveratrol;Calyculin A;LMPTP inhibitor 1 dihydrochloride;[pTyr5] EGFR (988-993) (TFA);RMC-3943;IKK-IN-3;AS1949490;PGAM1-IN-1;TD52 dihydrochloride;Daidzein-d4;Ciglitazone;bpV(phen)

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