R 59-022

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R 59-022

CAS No. : 93076-89-2

Biological Activity：R 59-022 (DKGI-I) is a diacylglycerol kinase inhibitor (IC50=2.8 μM). R 59-022 is a 5-HTR antagonist, and activates protein kinase C (PKC). R 59-022 potentiates thrombin-induced diacylglycerol production in platelets and inhibits phosphatidic acid production in neutrophils[2][3][4].

Research Area：Inflammation/Immunology

Targets：5-HT Receptor|PKC

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Related Small Molecules:F 13714;[Ala107]MBP(104-118) TFA;Mosapride-d5;BJE6-106;Myelin Basic Protein;Staurosporine;PKC-iota inhibitor 1;Nuciferine;Renzapride;Hypericin;LY 344864 racemate;Malantide;PKCiota-IN-2 formic;Harmine hydrochloride;Valerenic acid;Arotinolol;Melitracen-d6 hydrochloride;WAY-100635;Nelotanserin;Flupentixol-d4 dihydrochloride

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