PD 168368

For research use only. We do not sell to patients.

PD 168368

CAS No. : 204066-82-0

Biological Activity:PD 168368 is a potent, competitive, and selective neuromedin B receptor (NMB-R) antagonist with the Ki of 15–45 nM. PD 168368 is neuromedin B receptor (NMBR; IC50=96 nM) / gastrin-releasing peptide receptor (GRPR IC50=3500 nM) antagonist[2]. PD 168368 also is a mixed FPR1/FPR2/FPR3 agonist with EC50s of 0.57, 0.24, and 2.7 nM, respectively[3].

Research Area:Cancer

Targets:Bombesin Receptor

Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Anti-Cancer Compound Library;Anti-Breast Cancer Compound Library;

Related Small Molecules:PD176252;Bombesin;RC-3095;BA 1;BIM-26226;ML-18;Kuwanon H;MK-5046;Litorin;Ranatensin;Kuwanon G

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