Tag: Antagonist

For research use only. We do not sell to patients. ANQ-11125 TFA Biological Activity：ANQ-11125 TFA is a potent and selective antagonist of motilin, with the pKd of 8.24. ANQ-11125 TFA blocks motilide-induced contractions in vitro in the rabbit[2]. Research Area：Metabolic Disease Targets：Motilin Receptor Related Small Molecules:[Nle13]-Motilin;Camicinal;EM574;MA-2029;Motilin (26-47), human, porcine;DS-3801b Trending products：Recombinant Proteins  |  Bioactive Screening […]

For research use only. We do not sell to patients. Promethazine-d6 hydrochloride CAS No. : 1189947-02-1 Biological Activity：Promethazine-d6 ((±)-Promethazine-d6) hydrochloride is the deuterium labeled Promethazine hydrochloride. Promethazine hydrochloride is an orally active histamine receptor antagonist[2]. Research Area：Neurological Disease Targets：Histamine Receptor Related Small Molecules:Tripelennamine;Brompheniramine-d6 maleate;Samelisant;Chlorphenoxamine;H3 receptor-MO-1;Diphenhydramine;ABT-239;Ketotifen fumarate;Ranitidine;Cetirizine;Diphenylpyraline hydrochloride;Loratadine-d5;Phenyltoloxamine;Ritanserin;BMY-25271;FRG8701;Mecamylamine hydrochloride;Cimetidine sulfoxide;Brompheniramine maleate;Tecastemizole;Famotidine-13C,d3;Bromazine-d6 hydrochloride Trending products：Recombinant Proteins  |  […]

For research use only. We do not sell to patients. G907 CAS No. : 2244035-16-1 Biological Activity：G907 is a selective antagonist of ATP-binding cassette (ABC) transporter MsbA with anti-microbial activity. G907 inhibits E. coli MsbA with an IC50 value of 18 nM. G907 traps MsbA in an inward-facing, lipopolysaccharide-bound conformation by wedging into an architecturally […]

For research use only. We do not sell to patients. Veralipride CAS No. : 66644-81-3 Biological Activity：Veralipride is a D2 receptor antagonist. It is an alternative antidopaminergic treatment for menopausal symptoms. Research Area：Neurological Disease Targets：Dopamine Receptor Related Screening Libraries:Bioactive Compound Library Plus;GPCR/G Protein Compound Library;Neuronal Signaling Compound Library;Neurotransmitter Receptor Compound Library;Neurodegenerative Disease-related Compound Library;Human Metabolite […]

For research use only. We do not sell to patients. NMDA receptor antagonist 5 CAS No. : 2415998-36-4 Biological Activity：NMDA receptor antagonist 5 (Compound 10e) is a potent, brain permeable and non-toxic NMDA receptor antagonist. NMDA receptor antagonist 5 can be used for neurological disorder research. Research Area：Neurological Disease Targets：iGluR Related Small Molecules:CIQ;Quinolinic acid-d3;1-Aminocyclobutanecarboxylic acid;Glycine-1-13C,15N;ZL006;PYD-106;NMDA-IN-2;JAMI1001A;(S)-Willardiine;Fanapanel;(S)-AMPA;L-Glutamic […]

For research use only. We do not sell to patients. UT-155 CAS No. : 2031161-35-8 Biological Activity：UT-155 is a selective and potent androgen receptor (AR) antagonist, with a Ki of 267 nM for UT-155 binding to AR-LBD. Research Area：Cancer Targets：Androgen Receptor Related Screening Libraries:Bioactive Compound Library Plus;Anti-Cancer Compound Library;Transcription Factor-Targeted Library;Anti-Prostate Cancer Compound Library;Nuclear Receptor […]

For research use only. We do not sell to patients. Scyllatoxin CAS No. : 142948-19-4 Biological Activity：Scyllatoxin (Leiurotoxin I) is a peptide toxin, it can be isolated from the venom of the scorpion (Leiurus quinquestriatus hebraeus). Scyllatoxin is a blocker of small-conductance KCa (SK) channel. Scyllatoxin enhances both norepinephrine (NE) and epinephrine (Epi) release in […]

For research use only. We do not sell to patients. L-368,899 hydrochloride CAS No. : 160312-62-9 Biological Activity：L-368,899 hydrochloride is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptor, respectively. L-368,899 hydrochloride used as a tocolytic agent. Research Area：Endocrinology […]

For research use only. We do not sell to patients. (rel)-Asperparaline A CAS No. : 195966-93-9 Biological Activity：(rel)-Asperparaline A ((rel)-Aspergillimide), an anthelmintic metabolite, is isolated from okara that has been fermented with Aspergillus japonicas JV-23. (rel)-Asperparaline A is also a potent and selective antagonist of nAChR. (rel)-Asperparaline A exhibits paralytic activity in silk worms[2]. Research […]

For research use only. We do not sell to patients. Lintopride CAS No. : 107429-63-0 Biological Activity：Lintopride is a 5HT4 antagonist with moderate 5HT3 antagonist properties. Research Area：Neurological Disease Targets：5-HT Receptor Related Small Molecules:F 13714;Mosapride-d5;Nuciferine;Renzapride;LY 344864 racemate;Harmine hydrochloride;Valerenic acid;Arotinolol;Melitracen-d6 hydrochloride;WAY-100635;Nelotanserin;Flupentixol-d4 dihydrochloride;Cariprazine-d6 hydrochloride;Tetrahydro-β-carboline;CP-809101;Volinanserin-d4 hydrochloride;Masupirdine free base;BRL-15572 dihydrochloride;LY393558;Brexpiprazole S-oxide Trending products：Recombinant Proteins  |  Bioactive Screening Libraries  |  […]