EST73502

For research use only. We do not sell to patients.

EST73502

CAS No. : 1838622-25-5

Biological Activity:EST73502 is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 has antinociceptive activity.

Research Area:Neurological Disease

Targets:Opioid Receptor|Sigma Receptor

Related Small Molecules:ORL1 antagonist 1;Loperamide-d6 N-Oxide;Deltorphin 2 TFA;Nalfurafine;BD1063 dhydrochloride;β-Lipotropin (60-65);GSK1521498 free base;Trimebutine-d5 fumarate;Dynorphin B (1-13) (TFA);Dermorphin Analog;β-Endorphin (6-31), human;Phenyltoloxamine;JTC-801;E1R;Valorphin;Corydaline;TAN-452;Matrine;Naloxonazine dihydrochloride;[Leu5]-Enkephalin;Sec-O-Glucosylhamaudol;DPDPE;CTOP;β-Endorphin, equine;(±)-Vesamicol hydrochloride;Sigma-LIGAND-1

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